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Pharmacokinetics and metabolism of SRX246: a potent and selective vasopressin 1a antagonist.
J Pharm Sci. 2013 Jun;102(6):2033-2043. doi: 10.1002/jps.23495. Epub 2013 Mar 7.
J Pharm Sci. 2013.
PMID: 23471831
Synthesis and evaluation of potent and selective human V1a receptor antagonists as potential ligands for PET or SPECT imaging.
Fabio K, Guillon C, Lacey CJ, Lu SF, Heindel ND, Ferris CF, Placzek M, Jones G, Brownstein MJ, Simon NG.
Fabio K, et al.
Bioorg Med Chem. 2012 Feb 1;20(3):1337-45. doi: 10.1016/j.bmc.2011.12.013. Epub 2011 Dec 20.
Bioorg Med Chem. 2012.
PMID: 22249122
Free PMC article.
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Vasopressin antagonists as anxiolytics and antidepressants: recent developments.
Simon NG, Guillon C, Fabio K, Heindel ND, Lu SF, Miller M, Ferris CF, Brownstein MJ, Garripa C, Koppel GA.
Simon NG, et al.
Recent Pat CNS Drug Discov. 2008 Jun;3(2):77-93. doi: 10.2174/157488908784534586.
Recent Pat CNS Drug Discov. 2008.
PMID: 18537767
Review.
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Azetidinones as vasopressin V1a antagonists.
Guillon CD, Koppel GA, Brownstein MJ, Chaney MO, Ferris CF, Lu SF, Fabio KM, Miller MJ, Heindel ND, Hunden DC, Cooper RD, Kaldor SW, Skelton JJ, Dressman BA, Clay MP, Steinberg MI, Bruns RF, Simon NG.
Guillon CD, et al.
Bioorg Med Chem. 2007 Mar 1;15(5):2054-80. doi: 10.1016/j.bmc.2006.12.031. Epub 2006 Dec 23.
Bioorg Med Chem. 2007.
PMID: 17234419
Free PMC article.
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