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New bioisosteric sulphur-containing choline kinase inhibitors with a tracked mode of action.
Eur J Med Chem. 2023 Jan 15;246:115003. doi: 10.1016/j.ejmech.2022.115003. Epub 2022 Dec 5.
Eur J Med Chem. 2023.
PMID: 36493617
Biological Evaluation of New Thienopyridinium and Thienopyrimidinium Derivatives as Human Choline Kinase Inhibitors.
Luque-Navarro PM, Mariotto E, Ballarotto M, Rubbini G, Aguilar-Troyano FJ, Fasiolo A, Torretta A, Parisini E, Macchiarulo A, Laso A, Marco C, Viola G, Carrasco-Jimenez MP, López-Cara LC.
Luque-Navarro PM, et al.
Pharmaceutics. 2022 Mar 27;14(4):715. doi: 10.3390/pharmaceutics14040715.
Pharmaceutics. 2022.
PMID: 35456549
Free PMC article.
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Anticancer Activity of the Choline Kinase Inhibitor PL48 Is Due to Selective Disruption of Choline Metabolism and Transport Systems in Cancer Cell Lines.
García-Molina P, Sola-Leyva A, Luque-Navarro PM, Laso A, Ríos-Marco P, Ríos A, Lanari D, Torretta A, Parisini E, López-Cara LC, Marco C, Carrasco-Jiménez MP.
García-Molina P, et al. Among authors: luque navarro pm.
Pharmaceutics. 2022 Feb 16;14(2):426. doi: 10.3390/pharmaceutics14020426.
Pharmaceutics. 2022.
PMID: 35214160
Free PMC article.
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New Compounds with Bioisosteric Replacement of Classic Choline Kinase Inhibitors Show Potent Antiplasmodial Activity.
Aguilar-Troyano FJ, Torretta A, Rubbini G, Fasiolo A, Luque-Navarro PM, Carrasco-Jimenez MP, Pérez-Moreno G, Bosch-Navarrete C, González-Pacanowska D, Parisini E, Lopez-Cara LC.
Aguilar-Troyano FJ, et al. Among authors: luque navarro pm.
Pharmaceutics. 2021 Nov 2;13(11):1842. doi: 10.3390/pharmaceutics13111842.
Pharmaceutics. 2021.
PMID: 34834257
Free PMC article.
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Anticancer and Structure Activity Relationship of Non-Symmetrical Choline Kinase Inhibitors.
Schiaffino-Ortega S, Mariotto E, Luque-Navarro PM, Kimatrai-Salvador M, Rios-Marco P, Hurtado-Guerrero R, Marco C, Carrasco-Jimenez MP, Viola G, López-Cara LC.
Schiaffino-Ortega S, et al. Among authors: luque navarro pm.
Pharmaceutics. 2021 Aug 29;13(9):1360. doi: 10.3390/pharmaceutics13091360.
Pharmaceutics. 2021.
PMID: 34575436
Free PMC article.
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Flow Synthesis of Biologically-Relevant Compound Libraries.
Luque Navarro PM, Lanari D.
Luque Navarro PM, et al.
Molecules. 2020 Feb 18;25(4):909. doi: 10.3390/molecules25040909.
Molecules. 2020.
PMID: 32085549
Free PMC article.
Review.
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