Lozach O - Search Results

1

Combined Virtual and Experimental Screening for CK1 Inhibitors Identifies a Modulator of p53 and Reveals Important Aspects of in Silico Screening Performance.

Myrianthopoulos V, Lozach O, Zareifi D, Alexopoulos L, Meijer L, Gorgoulis VG, Mikros E. Myrianthopoulos V, et al. Among authors: lozach o. Int J Mol Sci. 2017 Oct 6;18(10):2102. doi: 10.3390/ijms18102102. Int J Mol Sci. 2017. PMID: 28984824 Free PMC article.

2

A facile consensus ranking approach enhances virtual screening robustness and identifies a cell-active DYRK1α inhibitor.

Mavrogeni ME, Pronios F, Zareifi D, Vasilakaki S, Lozach O, Alexopoulos L, Meijer L, Myrianthopoulos V, Mikros E. Mavrogeni ME, et al. Among authors: lozach o. Future Med Chem. 2018 Oct;10(20):2411-2430. doi: 10.4155/fmc-2018-0198. Epub 2018 Oct 16. Future Med Chem. 2018. PMID: 30325204 Free PMC article.

3

Further investigation of Paprotrain: Towards the conception of selective and multi-targeted CNS kinase inhibitors.

Labrière C, Lozach O, Blairvacq M, Meijer L, Guillou C. Labrière C, et al. Among authors: lozach o. Eur J Med Chem. 2016 Nov 29;124:920-934. doi: 10.1016/j.ejmech.2016.08.069. Epub 2016 Aug 31. Eur J Med Chem. 2016. PMID: 27676471

4

Soluble 3',6-substituted indirubins with enhanced selectivity toward glycogen synthase kinase -3 alter circadian period.

Vougogiannopoulou K, Ferandin Y, Bettayeb K, Myrianthopoulos V, Lozach O, Fan Y, Johnson CH, Magiatis P, Skaltsounis AL, Mikros E, Meijer L. Vougogiannopoulou K, et al. Among authors: lozach o. J Med Chem. 2008 Oct 23;51(20):6421-31. doi: 10.1021/jm800648y. Epub 2008 Sep 25. J Med Chem. 2008. PMID: 18816110 Free PMC article.

5

Novel Inverse Binding Mode of Indirubin Derivatives Yields Improved Selectivity for DYRK Kinases.

Myrianthopoulos V, Kritsanida M, Gaboriaud-Kolar N, Magiatis P, Ferandin Y, Durieu E, Lozach O, Cappel D, Soundararajan M, Filippakopoulos P, Sherman W, Knapp S, Meijer L, Mikros E, Skaltsounis AL. Myrianthopoulos V, et al. Among authors: lozach o. ACS Med Chem Lett. 2013 Jan 10;4(1):22-26. doi: 10.1021/ml300207a. Epub 2012 Nov 1. ACS Med Chem Lett. 2013. PMID: 23336033 Free PMC article.

6

Rebeccamycin derivatives as dual DNA-damaging agents and potent checkpoint kinase 1 inhibitors.

Marminon C, Anizon F, Moreau P, Pfeiffer B, Pierré A, Golsteyn RM, Peixoto P, Hildebrand MP, David-Cordonnier MH, Lozach O, Meijer L, Prudhomme M. Marminon C, et al. Among authors: lozach o. Mol Pharmacol. 2008 Dec;74(6):1620-9. doi: 10.1124/mol.108.049346. Epub 2008 Sep 2. Mol Pharmacol. 2008. PMID: 18768386

7

Synthesis, biological evaluation and molecular modelling studies of 4-anilinoquinazoline derivatives as protein kinase inhibitors.

Waiker DK, Karthikeyan C, Poongavanam V, Kongsted J, Lozach O, Meijer L, Trivedi P. Waiker DK, et al. Among authors: lozach o. Bioorg Med Chem. 2014 Mar 15;22(6):1909-15. doi: 10.1016/j.bmc.2014.01.044. Epub 2014 Jan 31. Bioorg Med Chem. 2014. PMID: 24530227

8

Anticancer alkaloid lamellarins inhibit protein kinases.

Baunbaek D, Trinkler N, Ferandin Y, Lozach O, Ploypradith P, Rucirawat S, Ishibashi F, Iwao M, Meijer L. Baunbaek D, et al. Among authors: lozach o. Mar Drugs. 2008;6(4):514-27. doi: 10.3390/md20080026. Epub 2008 Oct 7. Mar Drugs. 2008. PMID: 19172192 Free PMC article.

9

Synthesis and biological evaluation of tetrahydro[1,4]diazepino[1,2-a]indol-1-ones as cyclin-dependent kinase inhibitors.

Putey A, Fournet G, Lozach O, Perrin L, Meijer L, Joseph B. Putey A, et al. Among authors: lozach o. Eur J Med Chem. 2014 Aug 18;83:617-29. doi: 10.1016/j.ejmech.2014.06.063. Epub 2014 Jun 28. Eur J Med Chem. 2014. PMID: 24998602

10

Synthesis of new pyridazino[4,5-b]indol-4-ones and pyridazin-3(2H)-one analogs as DYRK1A inhibitors.

Bruel A, Bénéteau R, Chabanne M, Lozach O, Le Guevel R, Ravache M, Bénédetti H, Meijer L, Logé C, Robert JM. Bruel A, et al. Among authors: lozach o. Bioorg Med Chem Lett. 2014 Nov 1;24(21):5037-40. doi: 10.1016/j.bmcl.2014.09.017. Epub 2014 Sep 16. Bioorg Med Chem Lett. 2014. PMID: 25248682

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

73 results

Search Page