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Table representation of search results timeline featuring number of search results per year.

Year Number of Results
2010 2
2011 3
2012 2
2013 2
2014 2
2015 1
2016 5
2017 3
2018 6
2019 5
2020 3
2021 5
2022 5
2023 9
2024 3

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49 results

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Page 1
Sigma-1 Receptor Inhibition Reduces Mechanical Allodynia and Modulate Neuroinflammation in Chronic Neuropathic Pain.
Denaro S, Pasquinucci L, Turnaturi R, Alberghina C, Longhitano L, Giallongo S, Costanzo G, Spoto S, Grasso M, Zappalà A, Li Volti G, Tibullo D, Vicario N, Parenti R, Parenti C. Denaro S, et al. Among authors: pasquinucci l. Mol Neurobiol. 2024 May;61(5):2672-2685. doi: 10.1007/s12035-023-03717-w. Epub 2023 Nov 3. Mol Neurobiol. 2024. PMID: 37922065 Free PMC article.
Discovery of a novel series of potent carbonic anhydrase inhibitors with selective affinity for μ Opioid receptor for Safer and long-lasting analgesia.
Angeli A, Micheli L, Turnaturi R, Pasquinucci L, Parenti C, Alterio V, Di Fiore A, De Simone G, Monti SM, Carta F, Di Cesare Mannelli L, Ghelardini C, Supuran CT. Angeli A, et al. Among authors: pasquinucci l. Eur J Med Chem. 2023 Nov 15;260:115783. doi: 10.1016/j.ejmech.2023.115783. Epub 2023 Aug 30. Eur J Med Chem. 2023. PMID: 37678143
Discovery of first novel sigma/HDACi dual-ligands with a potent in vitro antiproliferative activity.
Barbaraci C, di Giacomo V, Maruca A, Patamia V, Rocca R, Dichiara M, Di Rienzo A, Cacciatore I, Cataldi A, Balaha M, Rapino M, Zagni C, Zampieri D, Pasquinucci L, Parenti C, Amata E, Rescifina A, Alcaro S, Marrazzo A. Barbaraci C, et al. Among authors: pasquinucci l. Bioorg Chem. 2023 Nov;140:106794. doi: 10.1016/j.bioorg.2023.106794. Epub 2023 Aug 23. Bioorg Chem. 2023. PMID: 37659146 Free article.
Discovery of AD258 as a Sigma Receptor Ligand with Potent Antiallodynic Activity.
Dichiara M, Ambrosio FA, Lee SM, Ruiz-Cantero MC, Lombino J, Coricello A, Costa G, Shah D, Costanzo G, Pasquinucci L, Son KN, Cosentino G, González-Cano R, Marrazzo A, Aakalu VK, Cobos EJ, Alcaro S, Amata E. Dichiara M, et al. Among authors: pasquinucci l. J Med Chem. 2023 Aug 24;66(16):11447-11463. doi: 10.1021/acs.jmedchem.3c00959. Epub 2023 Aug 3. J Med Chem. 2023. PMID: 37535861 Free PMC article.
Synthesis, Computational Insights, and Evaluation of Novel Sigma Receptors Ligands.
Dichiara M, Ambrosio FA, Barbaraci C, González-Cano R, Costa G, Parenti C, Marrazzo A, Pasquinucci L, Cobos EJ, Alcaro S, Amata E. Dichiara M, et al. Among authors: pasquinucci l. ACS Chem Neurosci. 2023 May 17;14(10):1845-1858. doi: 10.1021/acschemneuro.3c00074. Epub 2023 May 8. ACS Chem Neurosci. 2023. PMID: 37155827 Free PMC article.
49 results