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Rational design, synthesis and biological profiling of new KDM4C inhibitors.
Bioorg Med Chem. 2020 Jan 1;28(1):115128. doi: 10.1016/j.bmc.2019.115128. Epub 2019 Nov 8.
Bioorg Med Chem. 2020.
PMID: 31784197
Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases.
Mammoliti O, Jansen K, El Bkassiny S, Palisse A, Triballeau N, Bucher D, Allart B, Jaunet A, Tricarico G, De Wachter M, Menet C, Blanc J, Letfus V, Rupčić R, Šmehil M, Poljak T, Coornaert B, Sonck K, Duys I, Waeckel L, Lecru L, Marsais F, Jagerschmidt C, Auberval M, Pujuguet P, Oste L, Borgonovi M, Wakselman E, Christophe T, Houvenaghel N, Jans M, Heckmann B, Sanière L, Brys R.
Mammoliti O, et al. Among authors: letfus v.
J Med Chem. 2021 Oct 14;64(19):14557-14586. doi: 10.1021/acs.jmedchem.1c01066. Epub 2021 Sep 28.
J Med Chem. 2021.
PMID: 34581584
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Investigating the barriers to bioavailability of macrolide antibiotics in the rat.
Padovan J, Ralić J, Letfus V, Milić A, Bencetić Mihaljević V.
Padovan J, et al. Among authors: letfus v.
Eur J Drug Metab Pharmacokinet. 2012 Sep;37(3):163-71. doi: 10.1007/s13318-011-0074-5. Epub 2011 Nov 24.
Eur J Drug Metab Pharmacokinet. 2012.
PMID: 22113743
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[7-day period in the number of hospitalizations for myocardial infarction in the East-Bohemian Region during 1971--1974].
Letfus V, Kopecký K, Klimes J.
Letfus V, et al.
Cesk Zdrav. 1978;26(12):531-9.
Cesk Zdrav. 1978.
PMID: 729086
Czech.
No abstract available.
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