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Altiratinib Inhibits Tumor Growth, Invasion, Angiogenesis, and Microenvironment-Mediated Drug Resistance via Balanced Inhibition of MET, TIE2, and VEGFR2.
Mol Cancer Ther. 2015 Sep;14(9):2023-34. doi: 10.1158/1535-7163.MCT-14-1105. Epub 2015 Aug 18.
Mol Cancer Ther. 2015.
PMID: 26285778
The Selective Tie2 Inhibitor Rebastinib Blocks Recruitment and Function of Tie2Hi Macrophages in Breast Cancer and Pancreatic Neuroendocrine Tumors.
Harney AS, Karagiannis GS, Pignatelli J, Smith BD, Kadioglu E, Wise SC, Hood MM, Kaufman MD, Leary CB, Lu WP, Al-Ani G, Chen X, Entenberg D, Oktay MH, Wang Y, Chun L, De Palma M, Jones JG, Flynn DL, Condeelis JS.
Harney AS, et al. Among authors: leary cb.
Mol Cancer Ther. 2017 Nov;16(11):2486-2501. doi: 10.1158/1535-7163.MCT-17-0241. Epub 2017 Aug 24.
Mol Cancer Ther. 2017.
PMID: 28838996
Free PMC article.
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Ripretinib (DCC-2618) Is a Switch Control Kinase Inhibitor of a Broad Spectrum of Oncogenic and Drug-Resistant KIT and PDGFRA Variants.
Smith BD, Kaufman MD, Lu WP, Gupta A, Leary CB, Wise SC, Rutkoski TJ, Ahn YM, Al-Ani G, Bulfer SL, Caldwell TM, Chun L, Ensinger CL, Hood MM, McKinley A, Patt WC, Ruiz-Soto R, Su Y, Telikepalli H, Town A, Turner BA, Vogeti L, Vogeti S, Yates K, Janku F, Abdul Razak AR, Rosen O, Heinrich MC, Flynn DL.
Smith BD, et al. Among authors: leary cb.
Cancer Cell. 2019 May 13;35(5):738-751.e9. doi: 10.1016/j.ccell.2019.04.006.
Cancer Cell. 2019.
PMID: 31085175
Free article.
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Vimseltinib: A Precision CSF1R Therapy for Tenosynovial Giant Cell Tumors and Diseases Promoted by Macrophages.
Smith BD, Kaufman MD, Wise SC, Ahn YM, Caldwell TM, Leary CB, Lu WP, Tan G, Vogeti L, Vogeti S, Wilky BA, Davis LE, Sharma M, Ruiz-Soto R, Flynn DL.
Smith BD, et al. Among authors: leary cb.
Mol Cancer Ther. 2021 Nov;20(11):2098-2109. doi: 10.1158/1535-7163.MCT-21-0361. Epub 2021 Aug 25.
Mol Cancer Ther. 2021.
PMID: 34433663
Free PMC article.
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Discovery of vimseltinib (DCC-3014), a highly selective CSF1R switch-control kinase inhibitor, in clinical development for the treatment of Tenosynovial Giant Cell Tumor (TGCT).
Caldwell TM, Ahn YM, Bulfer SL, Leary CB, Hood MM, Lu WP, Vogeti L, Vogeti S, Kaufman MD, Wise SC, Le Bourdonnec B, Smith BD, Flynn DL.
Caldwell TM, et al. Among authors: leary cb.
Bioorg Med Chem Lett. 2022 Oct 15;74:128928. doi: 10.1016/j.bmcl.2022.128928. Epub 2022 Aug 10.
Bioorg Med Chem Lett. 2022.
PMID: 35961460
Free article.
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Selective dendrite-targeting of mRNAs of NR1 splice variants without exon 5: identification of a cis-acting sequence and isolation of sequence-binding proteins.
Pal R, Agbas A, Bao X, Hui D, Leary C, Hunt J, Naniwadekar A, Michaelis ML, Kumar KN, Michaelis EK.
Pal R, et al.
Brain Res. 2003 Dec 19;994(1):1-18. doi: 10.1016/j.brainres.2003.08.046.
Brain Res. 2003.
PMID: 14642443
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Factors Contributing to Early Intervention Evaluation.
Chan G, Gaither JR, Leventhal JM, Leary CB, Fenick AM.
Chan G, et al. Among authors: leary cb.
Acad Pediatr. 2022 Mar;22(2):227-232. doi: 10.1016/j.acap.2021.03.010. Epub 2021 Mar 18.
Acad Pediatr. 2022.
PMID: 33746044
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Use of nursing process to develop unit specific quality assurance plans.
Leary CB.
Leary CB.
J Nurs Qual Assur. 1990 Feb;4(2):1-6.
J Nurs Qual Assur. 1990.
PMID: 2312657
No abstract available.
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