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Synthesis, in vitro and in vivo giardicidal activity of nitrothiazole-NSAID chimeras displaying broad antiprotozoal spectrum.
Colín-Lozano B, León-Rivera I, Chan-Bacab MJ, Ortega-Morales BO, Moo-Puc R, López-Guerrero V, Hernández-Núñez E, Argüello-Garcia R, Scior T, Barbosa-Cabrera E, Navarrete-Vázquez G. Colín-Lozano B, et al. Bioorg Med Chem Lett. 2017 Aug 1;27(15):3490-3494. doi: 10.1016/j.bmcl.2017.05.071. Epub 2017 May 24. Bioorg Med Chem Lett. 2017. PMID: 28645659
Antidiabetic and toxicological evaluations of naringenin in normoglycaemic and NIDDM rat models and its implications on extra-pancreatic glucose regulation.
Ortiz-Andrade RR, Sánchez-Salgado JC, Navarrete-Vázquez G, Webster SP, Binnie M, García-Jiménez S, León-Rivera I, Cigarroa-Vázquez P, Villalobos-Molina R, Estrada-Soto S. Ortiz-Andrade RR, et al. Diabetes Obes Metab. 2008 Nov;10(11):1097-104. doi: 10.1111/j.1463-1326.2008.00869.x. Epub 2008 Mar 18. Diabetes Obes Metab. 2008. PMID: 18355329
Antidiabetic activity of N-(6-substituted-1,3-benzothiazol-2-yl)benzenesulfonamides.
Moreno-Díaz H, Villalobos-Molina R, Ortiz-Andrade R, Díaz-Coutiño D, Medina-Franco JL, Webster SP, Binnie M, Estrada-Soto S, Ibarra-Barajas M, León-Rivera I, Navarrete-Vázquez G. Moreno-Díaz H, et al. Bioorg Med Chem Lett. 2008 May 1;18(9):2871-7. doi: 10.1016/j.bmcl.2008.03.086. Epub 2008 Apr 8. Bioorg Med Chem Lett. 2008. PMID: 18424136
Design, synthesis and in vitro antiprotozoal activity of benzimidazole-pentamidine hybrids.
Torres-Gómez H, Hernández-Núñez E, León-Rivera I, Guerrero-Alvarez J, Cedillo-Rivera R, Moo-Puc R, Argotte-Ramos R, Rodríguez-Gutiérrez Mdel C, Chan-Bacab MJ, Navarrete-Vázquez G. Torres-Gómez H, et al. Bioorg Med Chem Lett. 2008 Jun 1;18(11):3147-51. doi: 10.1016/j.bmcl.2008.05.009. Epub 2008 May 4. Bioorg Med Chem Lett. 2008. PMID: 18486471
Synthesis, in vitro and computational studies of protein tyrosine phosphatase 1B inhibition of a small library of 2-arylsulfonylaminobenzothiazoles with antihyperglycemic activity.
Navarrete-Vazquez G, Paoli P, León-Rivera I, Villalobos-Molina R, Medina-Franco JL, Ortiz-Andrade R, Estrada-Soto S, Camici G, Diaz-Coutiño D, Gallardo-Ortiz I, Martinez-Mayorga K, Moreno-Díaz H. Navarrete-Vazquez G, et al. Bioorg Med Chem. 2009 May 1;17(9):3332-41. doi: 10.1016/j.bmc.2009.03.042. Epub 2009 Mar 26. Bioorg Med Chem. 2009. PMID: 19362487
Synthesis, vasorelaxant activity and antihypertensive effect of benzo[d]imidazole derivatives.
Navarrete-Vázquez G, Hidalgo-Figueroa S, Torres-Piedra M, Vergara-Galicia J, Rivera-Leyva JC, Estrada-Soto S, León-Rivera I, Aguilar-Guardarrama B, Rios-Gómez Y, Villalobos-Molina R, Ibarra-Barajas M. Navarrete-Vázquez G, et al. Bioorg Med Chem. 2010 Jun 1;18(11):3985-91. doi: 10.1016/j.bmc.2010.04.027. Epub 2010 Apr 14. Bioorg Med Chem. 2010. PMID: 20451399
Design, synthesis, and in vitro antiprotozoal, antimycobacterial activities of N-{2-[(7-chloroquinolin-4-yl)amino]ethyl}ureas.
Nava-Zuazo C, Estrada-Soto S, Guerrero-Alvarez J, León-Rivera I, Molina-Salinas GM, Said-Fernández S, Chan-Bacab MJ, Cedillo-Rivera R, Moo-Puc R, Mirón-López G, Navarrete-Vazquez G. Nava-Zuazo C, et al. Bioorg Med Chem. 2010 Sep 1;18(17):6398-403. doi: 10.1016/j.bmc.2010.07.008. Epub 2010 Jul 30. Bioorg Med Chem. 2010. PMID: 20674375
43 results