Lacivita E - Search Results

1

International Union of Basic and Clinical Pharmacology. CX. Classification of Receptors for 5-hydroxytryptamine; Pharmacology and Function.

Barnes NM, Ahern GP, Becamel C, Bockaert J, Camilleri M, Chaumont-Dubel S, Claeysen S, Cunningham KA, Fone KC, Gershon M, Di Giovanni G, Goodfellow NM, Halberstadt AL, Hartley RM, Hassaine G, Herrick-Davis K, Hovius R, Lacivita E, Lambe EK, Leopoldo M, Levy FO, Lummis SCR, Marin P, Maroteaux L, McCreary AC, Nelson DL, Neumaier JF, Newman-Tancredi A, Nury H, Roberts A, Roth BL, Roumier A, Sanger GJ, Teitler M, Sharp T, Villalón CM, Vogel H, Watts SW, Hoyer D. Barnes NM, et al. Among authors: lacivita e. Pharmacol Rev. 2021 Jan;73(1):310-520. doi: 10.1124/pr.118.015552. Pharmacol Rev. 2021. PMID: 33370241 Free PMC article. Review.

2

Structure-affinity relationship study on N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D(3) receptor ligands.

Leopoldo M, Berardi F, Colabufo NA, De Giorgio P, Lacivita E, Perrone R, Tortorella V. Leopoldo M, et al. Among authors: lacivita e. J Med Chem. 2002 Dec 19;45(26):5727-35. doi: 10.1021/jm020952a. J Med Chem. 2002. PMID: 12477356

3

Synthesis and structure-affinity relationships of 1-[omega-(4-aryl-1-piperazinyl)alkyl]-1-aryl ketones as 5-HT(7) receptor ligands.

Perrone R, Berardi F, Colabufo NA, Lacivita E, Leopoldo M, Tortorella V. Perrone R, et al. Among authors: lacivita e. J Med Chem. 2003 Feb 13;46(4):646-9. doi: 10.1021/jm020994z. J Med Chem. 2003. PMID: 12570387

4

Structure-affinity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agents.

Leopoldo M, Berardi F, Colabufo NA, Contino M, Lacivita E, Niso M, Perrone R, Tortorella V. Leopoldo M, et al. Among authors: lacivita e. J Med Chem. 2004 Dec 16;47(26):6616-24. doi: 10.1021/jm049702f. J Med Chem. 2004. PMID: 15588097

5

11C-labeling of n-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors.

Turolla EA, Matarrese M, Belloli S, Moresco RM, Simonelli P, Todde S, Fazio F, Magni F, Kienle MG, Leopoldo M, Berardi F, Colabufo NA, Lacivita E, Perrone R. Turolla EA, et al. Among authors: lacivita e. J Med Chem. 2005 Nov 3;48(22):7018-23. doi: 10.1021/jm050171k. J Med Chem. 2005. PMID: 16250661

6

Synthesis and binding profile of constrained analogues of N-[4-(4-arylpiperazin-1-yl)butyl]-3-methoxybenzamides, a class of potent dopamine D3 receptor ligands.

Leopoldo M, Lacivita E, Colabufo NA, Berardi F, Perrone R. Leopoldo M, et al. Among authors: lacivita e. J Pharm Pharmacol. 2006 Feb;58(2):209-18. doi: 10.1211/jpp.58.2.0008. J Pharm Pharmacol. 2006. PMID: 16451749

7

Selective agents for serotonin2C (5-HT2C) receptor.

Lacivita E, Leopoldo M. Lacivita E, et al. Curr Top Med Chem. 2006;6(18):1927-70. doi: 10.2174/156802606778522168. Curr Top Med Chem. 2006. PMID: 17017967 Review.

8

Bivalent ligand approach on 4-[2-(3-methoxyphenyl)ethyl]-1-(2-methoxyphenyl)piperazine: synthesis and binding affinities for 5-HT(7) and 5-HT(1A) receptors.

Leopoldo M, Lacivita E, Colabufo NA, Niso M, Berardi F, Perrone R. Leopoldo M, et al. Among authors: lacivita e. Bioorg Med Chem. 2007 Aug 1;15(15):5316-21. doi: 10.1016/j.bmc.2007.05.010. Epub 2007 May 6. Bioorg Med Chem. 2007. PMID: 17517509

9

Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinehexanamides, a class of 5-HT7 receptor agents. 2.

Leopoldo M, Lacivita E, Contino M, Colabufo NA, Berardi F, Perrone R. Leopoldo M, et al. Among authors: lacivita e. J Med Chem. 2007 Aug 23;50(17):4214-21. doi: 10.1021/jm070487n. Epub 2007 Jul 25. J Med Chem. 2007. PMID: 17649988

10

N-[omega-[4-(2-methoxyphenyl)-1-piperazinyl]alkyl]-2-quinolinamines as high-affinity fluorescent 5-HT1A receptor ligands.

Lacivita E, Leopoldo M. Lacivita E, et al. J Med Chem. 2008 Mar 13;51(5):1492-5. doi: 10.1021/jm7013919. Epub 2008 Feb 13. J Med Chem. 2008. PMID: 18269229

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