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IRAK4 inhibition dampens pathogenic processes driving inflammatory skin diseases.
Sci Transl Med. 2023 Feb 15;15(683):eabj3289. doi: 10.1126/scitranslmed.abj3289. Epub 2023 Feb 15.
Sci Transl Med. 2023.
PMID: 36791209
Discovery of 9-Cyclopropylethynyl-2-((S)-1-[1,4]dioxan-2-ylmethoxy)-6,7-dihydropyrimido[6,1-a]isoquinolin-4-one (GLPG1205), a Unique GPR84 Negative Allosteric Modulator Undergoing Evaluation in a Phase II Clinical Trial.
Labéguère F, Dupont S, Alvey L, Soulas F, Newsome G, Tirera A, Quenehen V, Mai TTT, Deprez P, Blanqué R, Oste L, Le Tallec S, De Vos S, Hagers A, Vandevelde A, Nelles L, Vandervoort N, Conrath K, Christophe T, van der Aar E, Wakselman E, Merciris D, Cottereaux C, da Costa C, Saniere L, Clement-Lacroix P, Jenkins L, Milligan G, Fletcher S, Brys R, Gosmini R.
Labéguère F, et al.
J Med Chem. 2020 Nov 25;63(22):13526-13545. doi: 10.1021/acs.jmedchem.0c00272. Epub 2020 Sep 23.
J Med Chem. 2020.
PMID: 32902984
Free article.
Clinical Trial.
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Three classes of ligands each bind to distinct sites on the orphan G protein-coupled receptor GPR84.
Mahmud ZA, Jenkins L, Ulven T, Labéguère F, Gosmini R, De Vos S, Hudson BD, Tikhonova IG, Milligan G.
Mahmud ZA, et al. Among authors: labeguere f.
Sci Rep. 2017 Dec 20;7(1):17953. doi: 10.1038/s41598-017-18159-3.
Sci Rep. 2017.
PMID: 29263400
Free PMC article.
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