TAK-137, an AMPA-R potentiator with little agonistic effect, has a wide therapeutic window.
Kunugi A, Tanaka M, Suzuki A, Tajima Y, Suzuki N, Suzuki M, Nakamura S, Kuno H, Yokota A, Sogabe S, Kosugi Y, Awasaki Y, Kaku T, Kimura H.
Kunugi A, et al.
Neuropsychopharmacology. 2019 Apr;44(5):961-970. doi: 10.1038/s41386-018-0213-7. Epub 2018 Sep 12.
Neuropsychopharmacology. 2019.
PMID: 30209408
Free PMC article.