Kristensen JL - Search Results

1

Discovery of β-Arrestin-Biased 25CN-NBOH-Derived 5-HT_2A Receptor Agonists.

Poulie CBM, Pottie E, Simon IA, Harpsøe K, D'Andrea L, Komarov IV, Gloriam DE, Jensen AA, Stove CP, Kristensen JL. Poulie CBM, et al. Among authors: kristensen jl. J Med Chem. 2022 Sep 22;65(18):12031-12043. doi: 10.1021/acs.jmedchem.2c00702. Epub 2022 Sep 13. J Med Chem. 2022. PMID: 36099411 Free PMC article.

2

N-Hydroxypyrazolyl glycine derivatives as selective N-methyl-D-aspartic acid receptor ligands.

Clausen RP, Christensen C, Hansen KB, Greenwood JR, Jørgensen L, Micale N, Madsen JC, Nielsen B, Egebjerg J, Bräuner-Osborne H, Traynelis SF, Kristensen JL. Clausen RP, et al. Among authors: kristensen jl. J Med Chem. 2008 Jul 24;51(14):4179-87. doi: 10.1021/jm800025e. Epub 2008 Jun 25. J Med Chem. 2008. PMID: 18578474 Free PMC article.

3

Novel 4-(piperidin-4-yl)-1-hydroxypyrazoles as gamma-aminobutyric acid(A) receptor ligands: synthesis, pharmacology, and structure-activity relationships.

Møller HA, Sander T, Kristensen JL, Nielsen B, Krall J, Bergmann ML, Christiansen B, Balle T, Jensen AA, Frølund B. Møller HA, et al. Among authors: kristensen jl. J Med Chem. 2010 Apr 22;53(8):3417-21. doi: 10.1021/jm100106r. J Med Chem. 2010. PMID: 20355712

4

Synthesis and biological evaluation of 4-(aminomethyl)-1-hydroxypyrazole analogues of muscimol as γ-aminobutyric acid(a) receptor agonists.

Petersen JG, Bergmann R, Møller HA, Jørgensen CG, Nielsen B, Kehler J, Frydenvang K, Kristensen J, Balle T, Jensen AA, Kristiansen U, Frølund B. Petersen JG, et al. J Med Chem. 2013 Feb 14;56(3):993-1006. doi: 10.1021/jm301473k. Epub 2013 Jan 23. J Med Chem. 2013. PMID: 23294161

5

Design, synthesis, and biological evaluation of Erythrina alkaloid analogues as neuronal nicotinic acetylcholine receptor antagonists.

Crestey F, Jensen AA, Borch M, Andreasen JT, Andersen J, Balle T, Kristensen JL. Crestey F, et al. Among authors: kristensen jl. J Med Chem. 2013 Dec 12;56(23):9673-82. doi: 10.1021/jm4013592. Epub 2013 Nov 21. J Med Chem. 2013. PMID: 24187998

6

Structure-activity relationships of constrained phenylethylamine ligands for the serotonin 5-HT2 receptors.

Isberg V, Paine J, Leth-Petersen S, Kristensen JL, Gloriam DE. Isberg V, et al. Among authors: kristensen jl. PLoS One. 2013 Nov 7;8(11):e78515. doi: 10.1371/journal.pone.0078515. eCollection 2013. PLoS One. 2013. PMID: 24244317 Free PMC article.

7

Synthesis and SAR study of a novel series of dopamine receptor agonists.

Risgaard R, Jensen M, Jørgensen M, Bang-Andersen B, Christoffersen CT, Jensen KG, Kristensen JL, Püschl A. Risgaard R, et al. Among authors: kristensen jl. Bioorg Med Chem. 2014 Jan 1;22(1):381-92. doi: 10.1016/j.bmc.2013.11.012. Epub 2013 Nov 15. Bioorg Med Chem. 2014. PMID: 24296012

8

Synthesis and structure-activity relationships of N-benzyl phenethylamines as 5-HT2A/2C agonists.

Hansen M, Phonekeo K, Paine JS, Leth-Petersen S, Begtrup M, Bräuner-Osborne H, Kristensen JL. Hansen M, et al. Among authors: kristensen jl. ACS Chem Neurosci. 2014 Mar 19;5(3):243-9. doi: 10.1021/cn400216u. Epub 2014 Jan 15. ACS Chem Neurosci. 2014. PMID: 24397362 Free PMC article.

9

Correlating the metabolic stability of psychedelic 5-HT₂A agonists with anecdotal reports of human oral bioavailability.

Leth-Petersen S, Bundgaard C, Hansen M, Carnerup MA, Kehler J, Kristensen JL. Leth-Petersen S, et al. Among authors: kristensen jl. Neurochem Res. 2014 Oct;39(10):2018-23. doi: 10.1007/s11064-014-1253-y. Epub 2014 Feb 12. Neurochem Res. 2014. PMID: 24519542

10

Synthesis and Pharmacological Evaluation of DHβE Analogues as Neuronal Nicotinic Acetylcholine Receptor Antagonists.

Jepsen TH, Jensen AA, Lund MH, Glibstrup E, Kristensen JL. Jepsen TH, et al. Among authors: kristensen jl. ACS Med Chem Lett. 2014 May 20;5(7):766-70. doi: 10.1021/ml500094c. eCollection 2014 Jul 10. ACS Med Chem Lett. 2014. PMID: 25050162 Free PMC article.

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