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New trifluoromethyl triazolopyrimidines as anti-Plasmodium falciparum agents.
Boechat N, Pinheiro LC, Silva TS, Aguiar AC, Carvalho AS, Bastos MM, Costa CC, Pinheiro S, Pinto AC, Mendonça JS, Dutra KD, Valverde AL, Santos-Filho OA, Ceravolo IP, Krettli AU. Boechat N, et al. Among authors: krettli au. Molecules. 2012 Jul 10;17(7):8285-302. doi: 10.3390/molecules17078285. Molecules. 2012. PMID: 22781441 Free PMC article.
Anti-Plasmodium falciparum activity of quinoline-sulfonamide hybrids.
Pinheiro LC, Boechat N, Ferreira Mde L, Júnior CC, Jesus AM, Leite MM, Souza NB, Krettli AU. Pinheiro LC, et al. Among authors: krettli au. Bioorg Med Chem. 2015 Sep 1;23(17):5979-84. doi: 10.1016/j.bmc.2015.06.056. Epub 2015 Jul 2. Bioorg Med Chem. 2015. PMID: 26190461
New hybrid trifluoromethylquinolines as antiplasmodium agents.
da Silva RMRJ, Gandi MO, Mendonça JS, Carvalho AS, Coutinho JP, Aguiar ACC, Krettli AU, Boechat N. da Silva RMRJ, et al. Among authors: krettli au. Bioorg Med Chem. 2019 Mar 15;27(6):1002-1008. doi: 10.1016/j.bmc.2019.01.044. Epub 2019 Feb 2. Bioorg Med Chem. 2019. PMID: 30737133 Free article.
MEFAS, a hybrid of artesunate-mefloquine active against asexual stages of Plasmodium vivax in field isolates, inhibits malaria transmission.
Penna-Coutinho J, da Silva Araújo M, Campos Aguiar AC, Sá PM, Rios CT, Medeiros JF, Pereira DB, Boechat N, Krettli AU. Penna-Coutinho J, et al. Among authors: krettli au. Int J Parasitol Drugs Drug Resist. 2021 Dec;17:150-155. doi: 10.1016/j.ijpddr.2021.09.003. Epub 2021 Sep 22. Int J Parasitol Drugs Drug Resist. 2021. PMID: 34637981 Free PMC article.
152 results