Krall J - Search Results

1

Pregnenolone sulfate analogues differentially modulate GABA_A receptor closed/desensitised states.

Mortensen M, Xu Y, Shehata MA, Krall J, Ernst M, Frølund B, Smart TG. Mortensen M, et al. Among authors: krall j. Br J Pharmacol. 2023 Oct;180(19):2482-2499. doi: 10.1111/bph.16143. Epub 2023 Jun 2. Br J Pharmacol. 2023. PMID: 37194503 Free PMC article.

2

GABAA receptor partial agonists and antagonists: structure, binding mode, and pharmacology.

Krall J, Balle T, Krogsgaard-Larsen N, Sørensen TE, Krogsgaard-Larsen P, Kristiansen U, Frølund B. Krall J, et al. Adv Pharmacol. 2015;72:201-27. doi: 10.1016/bs.apha.2014.10.003. Epub 2014 Dec 4. Adv Pharmacol. 2015. PMID: 25600372 Review.

3

Developing New 4-PIOL and 4-PHP Analogues for Photoinactivation of γ-Aminobutyric Acid Type A Receptors.

Mortensen M, Krall J, Kongstad KT, Brygger BM, Lenzi O, Francotte P, Sørensen TE, Nielsen B, Jensen AA, Smart TG, Frølund B. Mortensen M, et al. Among authors: krall j. ACS Chem Neurosci. 2019 Nov 20;10(11):4669-4684. doi: 10.1021/acschemneuro.9b00478. Epub 2019 Oct 21. ACS Chem Neurosci. 2019. PMID: 31589403

4

Silencing of spontaneous activity at α4β1/3δ GABA_A receptors in hippocampal granule cells reveals different ligand pharmacology.

Dalby NO, Falk-Petersen CB, Leurs U, Scholze P, Krall J, Frølund B, Wellendorph P. Dalby NO, et al. Among authors: krall j. Br J Pharmacol. 2020 Sep;177(17):3975-3990. doi: 10.1111/bph.15146. Epub 2020 Jul 15. Br J Pharmacol. 2020. PMID: 32484592 Free PMC article.

5

Discovery and Optimization of 5-Hydroxy-Diclofenac toward a New Class of Ligands with Nanomolar Affinity for the CaMKIIα Hub Domain.

Tian Y, Shehata MA, Gauger SJ, Ng CKL, Solbak S, Thiesen L, Bruus-Jensen J, Krall J, Bundgaard C, Gibson KM, Wellendorph P, Frølund B. Tian Y, et al. Among authors: krall j. J Med Chem. 2022 May 12;65(9):6656-6676. doi: 10.1021/acs.jmedchem.1c02177. Epub 2022 May 2. J Med Chem. 2022. PMID: 35500061

6

Exploring the orthosteric binding site of the γ-aminobutyric acid type A receptor using 4-(Piperidin-4-yl)-1-hydroxypyrazoles 3- or 5-imidazolyl substituted: design, synthesis, and pharmacological evaluation.

Krall J, Jensen CH, Sørensen TE, Nielsen B, Jensen AA, Sander T, Balle T, Frølund B. Krall J, et al. J Med Chem. 2013 Aug 22;56(16):6536-40. doi: 10.1021/jm4006466. Epub 2013 Aug 8. J Med Chem. 2013. PMID: 23855889

7

Probing α4βδ GABAA receptor heterogeneity: differential regional effects of a functionally selective α4β1δ/α4β3δ receptor agonist on tonic and phasic inhibition in rat brain.

Hoestgaard-Jensen K, Dalby NO, Krall J, Hammer H, Krogsgaard-Larsen P, Frølund B, Jensen AA. Hoestgaard-Jensen K, et al. Among authors: krall j. J Neurosci. 2014 Dec 3;34(49):16256-72. doi: 10.1523/JNEUROSCI.1495-14.2014. J Neurosci. 2014. PMID: 25471566 Free PMC article.

8

Imidazole-4-acetic acid, a new lead structure for interaction with the taurine transporter in outer blood-retinal barrier cells.

Valembois S, Krall J, Frølund B, Steffansen B. Valembois S, et al. Among authors: krall j. Eur J Pharm Sci. 2017 May 30;103:77-84. doi: 10.1016/j.ejps.2017.02.041. Epub 2017 Mar 1. Eur J Pharm Sci. 2017. PMID: 28259832

9

Sex-specific alterations in GABA receptor-mediated responses in laterodorsal tegmentum are associated with prenatal exposure to nicotine.

Eliasen JN, Krall J, Frølund B, Kohlmeier KA. Eliasen JN, et al. Among authors: krall j. Dev Neurobiol. 2020 May;80(5-6):178-199. doi: 10.1002/dneu.22772. Epub 2020 Aug 4. Dev Neurobiol. 2020. PMID: 32628361

10

Exploring the NCS-382 Scaffold for CaMKIIα Modulation: Synthesis, Biochemical Pharmacology, and Biophysical Characterization of Ph-HTBA as a Novel High-Affinity Brain-Penetrant Stabilizer of the CaMKIIα Hub Domain.

Tian Y, Shehata MA, Gauger SJ, Veronesi C, Hamborg L, Thiesen L, Bruus-Jensen J, Royssen JS, Leurs U, Larsen ASG, Krall J, Solbak SMØ, Wellendorph P, Frølund B. Tian Y, et al. Among authors: krall j. J Med Chem. 2022 Nov 24;65(22):15066-15084. doi: 10.1021/acs.jmedchem.2c00805. Epub 2022 Nov 8. J Med Chem. 2022. PMID: 36346645

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