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Page 1
Synthesis and biological evaluation of PSMA-targeting paclitaxel conjugates.
Machulkin AE, Skvortsov DA, Ivanenkov YA, Ber AP, Kavalchuk MV, Aladinskaya AV, Uspenskaya AA, Shafikov RR, Plotnikova EA, Yakubovskaya RI, Nimenko EA, Zyk NU, Beloglazkina EK, Zyk NV, Koteliansky VE, Majouga AG. Machulkin AE, et al. Among authors: koteliansky ve. Bioorg Med Chem Lett. 2019 Aug 15;29(16):2229-2235. doi: 10.1016/j.bmcl.2019.06.035. Epub 2019 Jun 20. Bioorg Med Chem Lett. 2019. PMID: 31248772
Synthesis, isomerization and biological activity of novel 2-selenohydantoin derivatives.
Ivanenkov YA, Veselov MS, Rezekin IG, Skvortsov DA, Sandulenko YB, Polyakova MV, Bezrukov DS, Vasilevsky SV, Kukushkin ME, Moiseeva AA, Finko AV, Koteliansky VE, Klyachko NL, Filatova LA, Beloglazkina EK, Zyk NV, Majouga AG. Ivanenkov YA, et al. Among authors: koteliansky ve. Bioorg Med Chem. 2016 Feb 15;24(4):802-11. doi: 10.1016/j.bmc.2015.12.050. Epub 2016 Jan 2. Bioorg Med Chem. 2016. PMID: 26780833
Small-molecule PSMA ligands. Current state, SAR and perspectives.
Machulkin AE, Ivanenkov YA, Aladinskaya AV, Veselov MS, Aladinskiy VA, Beloglazkina EK, Koteliansky VE, Shakhbazyan AG, Sandulenko YB, Majouga AG. Machulkin AE, et al. Among authors: koteliansky ve. J Drug Target. 2016 Sep;24(8):679-93. doi: 10.3109/1061186X.2016.1154564. Epub 2016 Mar 10. J Drug Target. 2016. PMID: 26887438 Review.
Synthesis and biological evaluation of Doxorubicin-containing conjugate targeting PSMA.
Ivanenkov YA, Machulkin AE, Garanina AS, Skvortsov DA, Uspenskaya AA, Deyneka EV, Trofimenko AV, Beloglazkina EK, Zyk NV, Koteliansky VE, Bezrukov DS, Aladinskaya AV, Vorobyeva NS, Puchinina MM, Riabykh GK, Sofronova AA, Malyshev AS, Majouga AG. Ivanenkov YA, et al. Among authors: koteliansky ve. Bioorg Med Chem Lett. 2019 May 15;29(10):1246-1255. doi: 10.1016/j.bmcl.2019.01.040. Epub 2019 Feb 1. Bioorg Med Chem Lett. 2019. PMID: 30904185
Corrigendum to 'Synthesis and biological evaluation of Doxorubicin-containing conjugate targeting PSMA' [Bioor. Med. Chem. Lett. 29/10 (2019) 1246-1255].
Ivanenkov YA, Machulkin AE, Garanina AS, Skvortsov DA, Uspenskaya AA, Deyneka EV, Trofimenko AV, Beloglazkina EK, Zyk NV, Koteliansky VE, Bezrukov DS, Aladinskaya AV, Vorobyeva NS, Puchinina MM, Ryabykh GK, Sofronova AA, Malyshev AS, Majouga AG. Ivanenkov YA, et al. Among authors: koteliansky ve. Bioorg Med Chem Lett. 2019 Jul 1;29(13):1688. doi: 10.1016/j.bmcl.2019.04.038. Epub 2019 May 2. Bioorg Med Chem Lett. 2019. PMID: 31056242 No abstract available.
In Silico Approaches to the Design of NS5A Inhibitors.
Ivanenkov YA, Veselov MS, Aladinskiy VA, Shakhbazyan AG, Yartseva SM, Majouga AG, Aladinskaya AV, Vantskul AS, Leonov SV, Ivachtchenko AV, Koteliansky VE. Ivanenkov YA, et al. Among authors: koteliansky ve. Curr Top Med Chem. 2016;16(12):1383-91. doi: 10.2174/1568026616666151120113705. Curr Top Med Chem. 2016. PMID: 26585932 Review.
Identification of Novel Small-Molecule ASGP-R Ligands.
Majouga AG, Ivanenkov YA, Veselov MS, Lopuhov AV, Maklakova SV, Beloglazkina EK, Binevski PV, Klyachko NL, Sandulenko YB, Galkina NY, Koteliansky VE. Majouga AG, et al. Among authors: koteliansky ve. Curr Drug Deliv. 2016;13(8):1303-1312. doi: 10.2174/1567201813666160719144651. Curr Drug Deliv. 2016. PMID: 27440073
Lipid-like materials for low-dose, in vivo gene silencing.
Love KT, Mahon KP, Levins CG, Whitehead KA, Querbes W, Dorkin JR, Qin J, Cantley W, Qin LL, Racie T, Frank-Kamenetsky M, Yip KN, Alvarez R, Sah DW, de Fougerolles A, Fitzgerald K, Koteliansky V, Akinc A, Langer R, Anderson DG. Love KT, et al. Proc Natl Acad Sci U S A. 2010 Feb 2;107(5):1864-9. doi: 10.1073/pnas.0910603106. Epub 2010 Jan 11. Proc Natl Acad Sci U S A. 2010. PMID: 20080679 Free PMC article.
mRNA-Based Therapeutics - Advances and Perspectives.
Sergeeva OV, Koteliansky VE, Zatsepin TS. Sergeeva OV, et al. Among authors: koteliansky ve. Biochemistry (Mosc). 2016 Jul;81(7):709-22. doi: 10.1134/S0006297916070075. Biochemistry (Mosc). 2016. PMID: 27449617 Free article. Review.
203 results