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Discovery of a novel class of inhaled dual pharmacology muscarinic antagonist and β2 agonist (MABA) for the treatment of chronic obstructive pulmonary disease (COPD).
Bioorg Med Chem Lett. 2021 Jun 1;41:127975. doi: 10.1016/j.bmcl.2021.127975. Epub 2021 Mar 19.
Bioorg Med Chem Lett. 2021.
PMID: 33753262
Discovery of Clinical Candidate CHF-6366: A Novel Super-soft Dual Pharmacology Muscarinic Antagonist and β2 Agonist (MABA) for the Inhaled Treatment of Respiratory Diseases.
Carzaniga L, Linney ID, Rizzi A, Delcanale M, Schmidt W, Knight CK, Pastore F, Miglietta D, Carnini C, Cesari N, Riccardi B, Mileo V, Venturi L, Moretti E, Blackaby WP, Patacchini R, Accetta A, Biagetti M, Bassani F, Tondelli M, Murgo A, Battipaglia L, Villetti G, Puccini P, Catinella S, Civelli M, Rancati F.
Carzaniga L, et al. Among authors: knight ck.
J Med Chem. 2022 Aug 11;65(15):10233-10250. doi: 10.1021/acs.jmedchem.2c00609. Epub 2022 Jul 28.
J Med Chem. 2022.
PMID: 35901125
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A novel series of 2,5-substituted tryptamine derivatives as vascular 5HT1B/1D receptor antagonists.
Moloney GP, Robertson AD, Martin GR, MacLennan S, Mathews N, Dodsworth S, Sang PY, Knight C, Glen R.
Moloney GP, et al.
J Med Chem. 1997 Jul 18;40(15):2347-62. doi: 10.1021/jm9605849.
J Med Chem. 1997.
PMID: 9240350
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Synthesis and serotonergic activity of substituted 2, N-benzylcarboxamido-5-(2-ethyl-1-dioxoimidazolidinyl)-N, N-dimethyltryptamine derivatives: novel antagonists for the vascular 5-HT(1B)-like receptor.
Moloney GP, Martin GR, Mathews N, Milne A, Hobbs H, Dodsworth S, Sang PY, Knight C, Williams M, Maxwell M, Glen RC.
Moloney GP, et al.
J Med Chem. 1999 Jul 15;42(14):2504-26. doi: 10.1021/jm9706325.
J Med Chem. 1999.
PMID: 10411472
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Household food insecurity and medication "scrimping" among US adults with diabetes.
Knight CK, Probst JC, Liese AD, Sercye E, Jones SJ.
Knight CK, et al.
Prev Med. 2016 Feb;83:41-5. doi: 10.1016/j.ypmed.2015.11.031. Epub 2015 Dec 4.
Prev Med. 2016.
PMID: 26656403
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Pectenotoxin-2 synthetic studies. 3. Assessment of the capacity for stereocontrolled cyclization to form the entire C1-C26 subunit based upon the double bond geometry across C15-C16.
O'Connor PD, Knight CK, Friedrich D, Peng X, Paquette LA.
O'Connor PD, et al. Among authors: knight ck.
J Org Chem. 2007 Mar 2;72(5):1747-54. doi: 10.1021/jo062513f. Epub 2007 Feb 2.
J Org Chem. 2007.
PMID: 17269830
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The imaging photopolarimeter experiment on pioneer 10.
Gehrels T, Coffeen D, Tomasko M, Doose L, Swindell W, Castillo N, Kendall J, Clements A, Hämeen-Anttila J, Knight CK, Blenman C, Baker R, Best G, Baker L.
Gehrels T, et al. Among authors: knight ck.
Science. 1974 Jan 25;183(4122):318-20. doi: 10.1126/science.183.4122.318.
Science. 1974.
PMID: 17821095
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