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A dual-acting 5-HT6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties.
Eur J Med Chem. 2020 Dec 15;208:112765. doi: 10.1016/j.ejmech.2020.112765. Epub 2020 Aug 22.
Eur J Med Chem. 2020.
PMID: 32949963
Overcoming undesirable hERG affinity by incorporating fluorine atoms: A case of MAO-B inhibitors derived from 1 H-pyrrolo-[3,2-c]quinolines.
Grychowska K, Olejarz-Maciej A, Blicharz K, Pietruś W, Karcz T, Kurczab R, Koczurkiewicz P, Doroz-Płonka A, Latacz G, Keeri AR, Piska K, Satała G, Pęgiel J, Trybała W, Jastrzębska-Więsek M, Bojarski AJ, Lamaty F, Partyka A, Walczak M, Krawczyk M, Malikowska-Racia N, Popik P, Zajdel P.
Grychowska K, et al. Among authors: keeri ar.
Eur J Med Chem. 2022 Jun 5;236:114329. doi: 10.1016/j.ejmech.2022.114329. Epub 2022 Mar 29.
Eur J Med Chem. 2022.
PMID: 35397400
Free article.
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Me2Zn-Mediated Catalytic Enantio- and Diastereoselective Addition of TosMIC to Ketones.
Keeri AR, Gualandi A, Mazzanti A, Lewinski J, Cozzi PG.
Keeri AR, et al.
Chemistry. 2015 Dec 21;21(52):18949-52. doi: 10.1002/chem.201504362. Epub 2015 Nov 23.
Chemistry. 2015.
PMID: 26549317
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