Kaiser M - Search Results

1

Discovery and Optimization of a Compound Series Active against Trypanosoma cruzi, the Causative Agent of Chagas Disease.

Harrison JR, Sarkar S, Hampton S, Riley J, Stojanovski L, Sahlberg C, Appelqvist P, Erath J, Mathan V, Rodriguez A, Kaiser M, Pacanowska DG, Read KD, Johansson NG, Gilbert IH. Harrison JR, et al. Among authors: kaiser m. J Med Chem. 2020 Mar 26;63(6):3066-3089. doi: 10.1021/acs.jmedchem.9b01852. Epub 2020 Mar 5. J Med Chem. 2020. PMID: 32134269

2

Analogues of thiolactomycin as potential antimalarial agents.

Jones SM, Urch JE, Kaiser M, Brun R, Harwood JL, Berry C, Gilbert IH. Jones SM, et al. Among authors: kaiser m. J Med Chem. 2005 Sep 22;48(19):5932-41. doi: 10.1021/jm049067d. J Med Chem. 2005. PMID: 16161997

3

Deoxyuridine triphosphate nucleotidohydrolase as a potential antiparasitic drug target.

Nguyen C, Kasinathan G, Leal-Cortijo I, Musso-Buendia A, Kaiser M, Brun R, Ruiz-Pérez LM, Johansson NG, González-Pacanowska D, Gilbert IH. Nguyen C, et al. Among authors: kaiser m. J Med Chem. 2005 Sep 22;48(19):5942-54. doi: 10.1021/jm050111e. J Med Chem. 2005. PMID: 16161998

4

Design, synthesis and evaluation of novel uracil amino acid conjugates for the inhibition of Trypanosoma cruzi dUTPase.

Mc Carthy OK, Schipani A, Buendía AM, Ruiz-Perez LM, Kaiser M, Brun R, Pacanowska DG, Gilbert IH. Mc Carthy OK, et al. Among authors: kaiser m. Bioorg Med Chem Lett. 2006 Jul 15;16(14):3809-12. doi: 10.1016/j.bmcl.2006.04.027. Epub 2006 May 3. Bioorg Med Chem Lett. 2006. PMID: 16677813

5

DNA binding affinity of bisguanidine and bis(2-aminoimidazoline) derivatives with in vivo antitrypanosomal activity.

Dardonville C, Barrett MP, Brun R, Kaiser M, Tanious F, Wilson WD. Dardonville C, et al. Among authors: kaiser m. J Med Chem. 2006 Jun 15;49(12):3748-52. doi: 10.1021/jm060295c. J Med Chem. 2006. PMID: 16759117 Free article.

6

Acyclic nucleoside analogues as inhibitors of Plasmodium falciparum dUTPase.

Nguyen C, Ruda GF, Schipani A, Kasinathan G, Leal I, Musso-Buendia A, Kaiser M, Brun R, Ruiz-Pérez LM, Sahlberg BL, Johansson NG, Gonzalez-Pacanowska D, Gilbert IH. Nguyen C, et al. Among authors: kaiser m. J Med Chem. 2006 Jul 13;49(14):4183-95. doi: 10.1021/jm060126s. J Med Chem. 2006. PMID: 16821778

7

Synthesis and biological evaluation of phosphate prodrugs of 4-phospho-D-erythronohydroxamic acid, an inhibitor of 6-phosphogluconate dehydrogenase.

Ruda GF, Alibu VP, Mitsos C, Bidet O, Kaiser M, Brun R, Barrett MP, Gilbert IH. Ruda GF, et al. Among authors: kaiser m. ChemMedChem. 2007 Aug;2(8):1169-80. doi: 10.1002/cmdc.200700040. ChemMedChem. 2007. PMID: 17615587 Free PMC article.

8

Quinuclidine derivatives as potential antiparasitics.

Cammerer SB, Jimenez C, Jones S, Gros L, Lorente SO, Rodrigues C, Rodrigues JC, Caldera A, Ruiz Perez LM, da Souza W, Kaiser M, Brun R, Urbina JA, Gonzalez Pacanowska D, Gilbert IH. Cammerer SB, et al. Among authors: kaiser m. Antimicrob Agents Chemother. 2007 Nov;51(11):4049-61. doi: 10.1128/AAC.00205-07. Epub 2007 Aug 20. Antimicrob Agents Chemother. 2007. PMID: 17709461 Free PMC article.

9

Synthesis and evaluation of antiparasitic activities of new 4-[5-(4-phenoxyphenyl)-2H-pyrazol-3-yl]morpholine derivatives.

Kuettel S, Zambon A, Kaiser M, Brun R, Scapozza L, Perozzo R. Kuettel S, et al. Among authors: kaiser m. J Med Chem. 2007 Nov 15;50(23):5833-9. doi: 10.1021/jm700938n. Epub 2007 Oct 20. J Med Chem. 2007. PMID: 17949068

10

Novel azabicyclo[3.2.2]nonane derivatives and their activities against Plasmodium falciparum K1 and Trypanosoma brucei rhodesiense.

Berger H, Weis R, Kaiser M, Brun R, Saf R, Seebacher W. Berger H, et al. Among authors: kaiser m. Bioorg Med Chem. 2008 Jun 15;16(12):6371-8. doi: 10.1016/j.bmc.2008.05.007. Epub 2008 May 7. Bioorg Med Chem. 2008. PMID: 18502136

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