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Year | Number of Results |
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2022 | 1 |
2023 | 3 |
2024 | 0 |
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Page 1
The incretin co-agonist tirzepatide requires GIPR for hormone secretion from human islets.
Nat Metab. 2023 Jun;5(6):945-954. doi: 10.1038/s42255-023-00811-0. Epub 2023 Jun 5.
Nat Metab. 2023.
PMID: 37277609
Free PMC article.
Hypothalamic and brainstem glucose-dependent insulinotropic polypeptide receptor neurons employ distinct mechanisms to affect feeding.
Adriaenssens A, Broichhagen J, de Bray A, Ast J, Hasib A, Jones B, Tomas A, Burgos NF, Woodward O, Lewis J, O'Flaherty E, El K, Cui C, Harada N, Inagaki N, Campbell J, Brierley D, Hodson DJ, Samms R, Gribble F, Reimann F.
Adriaenssens A, et al.
JCI Insight. 2023 May 22;8(10):e164921. doi: 10.1172/jci.insight.164921.
JCI Insight. 2023.
PMID: 37212283
Free PMC article.
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The ubiquitination status of the glucagon receptor determines signal bias.
Kaur S, Sokrat B, Capozzi ME, El K, Bai Y, Jazic A, Han B, Krishna Kumar K, D'Alessio DA, Campbell JE, Bouvier M, Shenoy SK.
Kaur S, et al.
J Biol Chem. 2023 May;299(5):104690. doi: 10.1016/j.jbc.2023.104690. Epub 2023 Apr 8.
J Biol Chem. 2023.
PMID: 37037304
Free PMC article.
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Discovery of a potent GIPR peptide antagonist that is effective in rodent and human systems.
Yang B, Gelfanov VM, El K, Chen A, Rohlfs R, DuBois B, Kruse Hansen AM, Perez-Tilve D, Knerr PJ, D'Alessio D, Campbell JE, Douros JD, Finan B.
Yang B, et al.
Mol Metab. 2022 Dec;66:101638. doi: 10.1016/j.molmet.2022.101638. Epub 2022 Nov 15.
Mol Metab. 2022.
PMID: 36400403
Free PMC article.
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