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Picomolar fluorescent probes for compound affinity determination to carbonic anhydrase IX expressed in live cancer cells.
Sci Rep. 2022 Oct 21;12(1):17644. doi: 10.1038/s41598-022-22436-1.
Sci Rep. 2022.
PMID: 36271018
Free PMC article.
Intrinsic thermodynamics of sulfonamide inhibitor binding to human carbonic anhydrases I and II.
Morkūnaitė V, Gylytė J, Zubrienė A, Baranauskienė L, Kišonaitė M, Michailovienė V, Juozapaitienė V, Todd MJ, Matulis D.
Morkūnaitė V, et al. Among authors: juozapaitiene v.
J Enzyme Inhib Med Chem. 2015 Apr;30(2):204-11. doi: 10.3109/14756366.2014.908291. Epub 2014 Apr 23.
J Enzyme Inhib Med Chem. 2015.
PMID: 24758348
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Discovery and characterization of novel selective inhibitors of carbonic anhydrase IX.
Dudutienė V, Matulienė J, Smirnov A, Timm DD, Zubrienė A, Baranauskienė L, Morkūnaite V, Smirnovienė J, Michailovienė V, Juozapaitienė V, Mickevičiūtė A, Kazokaitė J, Bakšytė S, Kasiliauskaitė A, Jachno J, Revuckienė J, Kišonaitė M, Pilipuitytė V, Ivanauskaitė E, Milinavičiūtė G, Smirnovas V, Petrikaitė V, Kairys V, Petrauskas V, Norvaišas P, Lingė D, Gibieža P, Capkauskaitė E, Zakšauskas A, Kazlauskas E, Manakova E, Gražulis S, Ladbury JE, Matulis D.
Dudutienė V, et al. Among authors: juozapaitiene v.
J Med Chem. 2014 Nov 26;57(22):9435-46. doi: 10.1021/jm501003k. Epub 2014 Nov 10.
J Med Chem. 2014.
PMID: 25358084
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Intrinsic thermodynamics of inhibitor binding to human carbonic anhydrase IX.
Linkuvienė V, Matulienė J, Juozapaitienė V, Michailovienė V, Jachno J, Matulis D.
Linkuvienė V, et al. Among authors: juozapaitiene v.
Biochim Biophys Acta. 2016 Apr;1860(4):708-18. doi: 10.1016/j.bbagen.2016.01.007. Epub 2016 Jan 18.
Biochim Biophys Acta. 2016.
PMID: 26794023
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Purification, enzymatic activity and inhibitor discovery for recombinant human carbonic anhydrase XIV.
Juozapaitienė V, Bartkutė B, Michailovienė V, Zakšauskas A, Baranauskienė L, Satkūnė S, Matulis D.
Juozapaitienė V, et al.
J Biotechnol. 2016 Dec 20;240:31-42. doi: 10.1016/j.jbiotec.2016.10.018. Epub 2016 Oct 20.
J Biotechnol. 2016.
PMID: 27773757
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Structure and mechanism of secondary sulfonamide binding to carbonic anhydrases.
Baronas D, Dudutienė V, Paketurytė V, Kairys V, Smirnov A, Juozapaitienė V, Vaškevičius A, Manakova E, Gražulis S, Zubrienė A, Matulis D.
Baronas D, et al. Among authors: juozapaitiene v.
Eur Biophys J. 2021 Oct;50(7):993-1011. doi: 10.1007/s00249-021-01561-1. Epub 2021 Jul 30.
Eur Biophys J. 2021.
PMID: 34328515
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Intrinsic thermodynamics of 4-substituted-2,3,5,6-tetrafluorobenzenesulfonamide binding to carbonic anhydrases by isothermal titration calorimetry.
Zubrienė A, Smirnovienė J, Smirnov A, Morkūnaitė V, Michailovienė V, Jachno J, Juozapaitienė V, Norvaišas P, Manakova E, Gražulis S, Matulis D.
Zubrienė A, et al. Among authors: juozapaitiene v.
Biophys Chem. 2015 Oct;205:51-65. doi: 10.1016/j.bpc.2015.05.009. Epub 2015 Jun 6.
Biophys Chem. 2015.
PMID: 26079542
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High-Affinity NIR-Fluorescent Inhibitors for Tumor Imaging via Carbonic Anhydrase IX.
Žvinys G, Petrosiute A, Zakšauskas A, Zubrienė A, Ščerbavičienė A, Kalnina Z, Čapkauskaitė E, Juozapaitienė V, Mickevičiu Tė A, Shubin K, Grincevičienė Š, Raišys S, Tars K, Matulienė J, Matulis D.
Žvinys G, et al. Among authors: juozapaitiene v.
Bioconjug Chem. 2024 May 15. doi: 10.1021/acs.bioconjchem.4c00144. Online ahead of print.
Bioconjug Chem. 2024.
PMID: 38750635
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