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Picomolar fluorescent probes for compound affinity determination to carbonic anhydrase IX expressed in live cancer cells.
Matulienė J, Žvinys G, Petrauskas V, Kvietkauskaitė A, Zakšauskas A, Shubin K, Zubrienė A, Baranauskienė L, Kačenauskaitė L, Kopanchuk S, Veiksina S, Paketurytė-Latvė V, Smirnovienė J, Juozapaitienė V, Mickevičiūtė A, Michailovienė V, Jachno J, Stravinskienė D, Sližienė A, Petrošiūtė A, Becker HM, Kazokaitė-Adomaitienė J, Yaromina A, Čapkauskaitė E, Rinken A, Dudutienė V, Dubois LJ, Matulis D. Matulienė J, et al. Among authors: juozapaitiene v. Sci Rep. 2022 Oct 21;12(1):17644. doi: 10.1038/s41598-022-22436-1. Sci Rep. 2022. PMID: 36271018 Free PMC article.
Discovery and characterization of novel selective inhibitors of carbonic anhydrase IX.
Dudutienė V, Matulienė J, Smirnov A, Timm DD, Zubrienė A, Baranauskienė L, Morkūnaite V, Smirnovienė J, Michailovienė V, Juozapaitienė V, Mickevičiūtė A, Kazokaitė J, Bakšytė S, Kasiliauskaitė A, Jachno J, Revuckienė J, Kišonaitė M, Pilipuitytė V, Ivanauskaitė E, Milinavičiūtė G, Smirnovas V, Petrikaitė V, Kairys V, Petrauskas V, Norvaišas P, Lingė D, Gibieža P, Capkauskaitė E, Zakšauskas A, Kazlauskas E, Manakova E, Gražulis S, Ladbury JE, Matulis D. Dudutienė V, et al. Among authors: juozapaitiene v. J Med Chem. 2014 Nov 26;57(22):9435-46. doi: 10.1021/jm501003k. Epub 2014 Nov 10. J Med Chem. 2014. PMID: 25358084
Intrinsic thermodynamics of inhibitor binding to human carbonic anhydrase IX.
Linkuvienė V, Matulienė J, Juozapaitienė V, Michailovienė V, Jachno J, Matulis D. Linkuvienė V, et al. Among authors: juozapaitiene v. Biochim Biophys Acta. 2016 Apr;1860(4):708-18. doi: 10.1016/j.bbagen.2016.01.007. Epub 2016 Jan 18. Biochim Biophys Acta. 2016. PMID: 26794023
Structure and mechanism of secondary sulfonamide binding to carbonic anhydrases.
Baronas D, Dudutienė V, Paketurytė V, Kairys V, Smirnov A, Juozapaitienė V, Vaškevičius A, Manakova E, Gražulis S, Zubrienė A, Matulis D. Baronas D, et al. Among authors: juozapaitiene v. Eur Biophys J. 2021 Oct;50(7):993-1011. doi: 10.1007/s00249-021-01561-1. Epub 2021 Jul 30. Eur Biophys J. 2021. PMID: 34328515
Intrinsic thermodynamics of 4-substituted-2,3,5,6-tetrafluorobenzenesulfonamide binding to carbonic anhydrases by isothermal titration calorimetry.
Zubrienė A, Smirnovienė J, Smirnov A, Morkūnaitė V, Michailovienė V, Jachno J, Juozapaitienė V, Norvaišas P, Manakova E, Gražulis S, Matulis D. Zubrienė A, et al. Among authors: juozapaitiene v. Biophys Chem. 2015 Oct;205:51-65. doi: 10.1016/j.bpc.2015.05.009. Epub 2015 Jun 6. Biophys Chem. 2015. PMID: 26079542
High-Affinity NIR-Fluorescent Inhibitors for Tumor Imaging via Carbonic Anhydrase IX.
Žvinys G, Petrosiute A, Zakšauskas A, Zubrienė A, Ščerbavičienė A, Kalnina Z, Čapkauskaitė E, Juozapaitienė V, Mickevičiu Tė A, Shubin K, Grincevičienė Š, Raišys S, Tars K, Matulienė J, Matulis D. Žvinys G, et al. Among authors: juozapaitiene v. Bioconjug Chem. 2024 May 15. doi: 10.1021/acs.bioconjchem.4c00144. Online ahead of print. Bioconjug Chem. 2024. PMID: 38750635