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Can Cysteine Protease Cross-Class Inhibitors Achieve Selectivity?
Cianni L, Feldmann CW, Gilberg E, Gütschow M, Juliano L, Leitão A, Bajorath J, Montanari CA. Cianni L, et al. Among authors: juliano l. J Med Chem. 2019 Dec 12;62(23):10497-10525. doi: 10.1021/acs.jmedchem.9b00683. Epub 2019 Aug 15. J Med Chem. 2019. PMID: 31361135 Review.
Non-peptidic cruzain inhibitors with trypanocidal activity discovered by virtual screening and in vitro assay.
Wiggers HJ, Rocha JR, Fernandes WB, Sesti-Costa R, Carneiro ZA, Cheleski J, da Silva AB, Juliano L, Cezari MH, Silva JS, McKerrow JH, Montanari CA. Wiggers HJ, et al. Among authors: juliano l. PLoS Negl Trop Dis. 2013 Aug 22;7(8):e2370. doi: 10.1371/journal.pntd.0002370. eCollection 2013. PLoS Negl Trop Dis. 2013. PMID: 23991231 Free PMC article.
Isomannide derivatives as new class of inhibitors for human kallikrein 7.
Freitas RF, Teixeira TS, Barros TG, Santos JA, Kondo MY, Juliano MA, Juliano L, Blaber M, Antunes OA, Abrahão O Jr, Pinheiro S, Muri EM, Puzer L. Freitas RF, et al. Among authors: juliano l, juliano ma. Bioorg Med Chem Lett. 2012 Oct 1;22(19):6072-5. doi: 10.1016/j.bmcl.2012.08.047. Epub 2012 Aug 21. Bioorg Med Chem Lett. 2012. PMID: 22959247
Poliovirus 3C proteinase inhibition by organotelluranes.
Gouvea IE, Santos JA, Burlandy FM, Tersariol IL, da Silva EE, Juliano MA, Juliano L, Cunha RL. Gouvea IE, et al. Among authors: juliano l, juliano ma. Biol Chem. 2011 Apr;392(6):587-91. doi: 10.1515/BC.2011.059. Epub 2011 Apr 27. Biol Chem. 2011. PMID: 21521074
Antitumor effect of chiral organotelluranes elicited in a murine melanoma model.
Paschoalin T, Martens AA, Omori ÁT, Pereira FV, Juliano L, Travassos LR, Machado-Santelli GM, Cunha RLOR. Paschoalin T, et al. Among authors: juliano l. Bioorg Med Chem. 2019 Jun 15;27(12):2537-2545. doi: 10.1016/j.bmc.2019.03.032. Epub 2019 Mar 21. Bioorg Med Chem. 2019. PMID: 30962115
453 results