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Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice.
Mock ED, Mustafa M, Gunduz-Cinar O, Cinar R, Petrie GN, Kantae V, Di X, Ogasawara D, Varga ZV, Paloczi J, Miliano C, Donvito G, van Esbroeck ACM, van der Gracht AMF, Kotsogianni I, Park JK, Martella A, van der Wel T, Soethoudt M, Jiang M, Wendel TJ, Janssen APA, Bakker AT, Donovan CM, Castillo LI, Florea BI, Wat J, van den Hurk H, Wittwer M, Grether U, Holmes A, van Boeckel CAA, Hankemeier T, Cravatt BF, Buczynski MW, Hill MN, Pacher P, Lichtman AH, van der Stelt M. Mock ED, et al. Among authors: janssen apa. Nat Chem Biol. 2020 Jun;16(6):667-675. doi: 10.1038/s41589-020-0528-7. Epub 2020 May 11. Nat Chem Biol. 2020. PMID: 32393901 Free PMC article.
Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474.
van Esbroeck ACM, Janssen APA, Cognetta AB 3rd, Ogasawara D, Shpak G, van der Kroeg M, Kantae V, Baggelaar MP, de Vrij FMS, Deng H, Allarà M, Fezza F, Lin Z, van der Wel T, Soethoudt M, Mock ED, den Dulk H, Baak IL, Florea BI, Hendriks G, De Petrocellis L, Overkleeft HS, Hankemeier T, De Zeeuw CI, Di Marzo V, Maccarrone M, Cravatt BF, Kushner SA, van der Stelt M. van Esbroeck ACM, et al. Among authors: janssen apa. Science. 2017 Jun 9;356(6342):1084-1087. doi: 10.1126/science.aaf7497. Science. 2017. PMID: 28596366 Free PMC article.
Two-step activity-based protein profiling of diacylglycerol lipase.
van Rooden EJ, Kreekel R, Hansen T, Janssen APA, van Esbroeck ACM, den Dulk H, van den Berg RJBHN, Codée JDC, van der Stelt M. van Rooden EJ, et al. Among authors: janssen apa. Org Biomol Chem. 2018 Jul 25;16(29):5250-5253. doi: 10.1039/c8ob01499j. Org Biomol Chem. 2018. PMID: 30004552
ABHD2 Inhibitor Identified by Activity-Based Protein Profiling Reduces Acrosome Reaction.
Baggelaar MP, den Dulk H, Florea BI, Fazio D, Bernabò N, Raspa M, Janssen APA, Scavizzi F, Barboni B, Overkleeft HS, Maccarrone M, van der Stelt M. Baggelaar MP, et al. Among authors: janssen apa. ACS Chem Biol. 2019 Oct 18;14(10):2295-2304. doi: 10.1021/acschembio.9b00640. Epub 2019 Oct 1. ACS Chem Biol. 2019. PMID: 31525885 Free PMC article.
ABHD2 Inhibitor Identified by Activity-Based Protein Profiling Reduces Acrosome Reaction.
Baggelaar MP, den Dulk H, Florea BI, Fazio D, Perruzza D, Bernabò N, Raspa M, Janssen APA, Scavizzi F, Barboni B, Overkleeft HS, Maccarrone M, van der Stelt M. Baggelaar MP, et al. Among authors: janssen apa. ACS Chem Biol. 2019 Dec 20;14(12):2943. doi: 10.1021/acschembio.9b00824. Epub 2019 Nov 7. ACS Chem Biol. 2019. PMID: 31697462 Free PMC article. No abstract available.
Bioorthogonal protein labelling enables the study of antigen processing of citrullinated and carbamylated auto-antigens.
van Leeuwen T, Araman C, Pieper Pournara L, Kampstra ASB, Bakkum T, Marqvorsen MHS, Nascimento CR, Groenewold GJM, van der Wulp W, Camps MGM, Janssen GMC, van Veelen PA, van Westen GJP, Janssen APA, Florea BI, Overkleeft HS, Ossendorp FA, Toes REM, van Kasteren SI. van Leeuwen T, et al. Among authors: janssen apa. RSC Chem Biol. 2021 Feb 23;2(3):855-862. doi: 10.1039/d1cb00009h. RSC Chem Biol. 2021. PMID: 34212151 Free PMC article.
18 results