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Generation of a mutator parasite to drive resistome discovery in Plasmodium falciparum.
Nat Commun. 2023 May 27;14(1):3059. doi: 10.1038/s41467-023-38774-1.
Nat Commun. 2023.
PMID: 37244916
Free PMC article.
Exploring a Tetrahydroquinoline Antimalarial Hit from the Medicines for Malaria Pathogen Box and Identification of its Mode of Resistance as PfeEF2.
Laleu B, Rubiano K, Yeo T, Hallyburton I, Anderson M, Crespo-Fernandez B, Gamo FJ, Antonova-Koch Y, Orjuela-Sanchez P, Wittlin S, Jana GP, Maity BC, Chenu E, Duffy J, Sjö P, Waterson D, Winzeler E, Guantai E, Fidock DA, Hansson TG.
Laleu B, et al. Among authors: jana gp.
ChemMedChem. 2022 Nov 18;17(22):e202200393. doi: 10.1002/cmdc.202200393. Epub 2022 Oct 13.
ChemMedChem. 2022.
PMID: 36129427
Free PMC article.
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Reaction hijacking inhibition of Plasmodium falciparum asparagine tRNA synthetase.
Xie SC, Wang Y, Morton CJ, Metcalfe RD, Dogovski C, Pasaje CFA, Dunn E, Luth MR, Kumpornsin K, Istvan ES, Park JS, Fairhurst KJ, Ketprasit N, Yeo T, Yildirim O, Bhebhe MN, Klug DM, Rutledge PJ, Godoy LC, Dey S, De Souza ML, Siqueira-Neto JL, Du Y, Puhalovich T, Amini M, Shami G, Loesbanluechai D, Nie S, Williamson N, Jana GP, Maity BC, Thomson P, Foley T, Tan DS, Niles JC, Han BW, Goldberg DE, Burrows J, Fidock DA, Lee MCS, Winzeler EA, Griffin MDW, Todd MH, Tilley L.
Xie SC, et al. Among authors: jana gp.
Res Sq [Preprint]. 2023 Jul 27:rs.3.rs-3198291. doi: 10.21203/rs.3.rs-3198291/v1.
Res Sq. 2023.
PMID: 37546892
Free PMC article.
Updated.
Preprint.
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Reaction hijacking inhibition of Plasmodium falciparum asparagine tRNA synthetase.
Xie SC, Wang Y, Morton CJ, Metcalfe RD, Dogovski C, Pasaje CFA, Dunn E, Luth MR, Kumpornsin K, Istvan ES, Park JS, Fairhurst KJ, Ketprasit N, Yeo T, Yildirim O, Bhebhe MN, Klug DM, Rutledge PJ, Godoy LC, Dey S, De Souza ML, Siqueira-Neto JL, Du Y, Puhalovich T, Amini M, Shami G, Loesbanluechai D, Nie S, Williamson N, Jana GP, Maity BC, Thomson P, Foley T, Tan DS, Niles JC, Han BW, Goldberg DE, Burrows J, Fidock DA, Lee MCS, Winzeler EA, Griffin MDW, Todd MH, Tilley L.
Xie SC, et al. Among authors: jana gp.
Nat Commun. 2024 Jan 31;15(1):937. doi: 10.1038/s41467-024-45224-z.
Nat Commun. 2024.
PMID: 38297033
Free PMC article.
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