Jacques Y. Roberge - Search Results

Year	Number of Results
2002	1
2004	2
2005	2
2009	1
2011	2
2013	1
2014	1
2021	3
2022	2
2023	1
2024	3

1

A FtsZ Inhibitor That Can Utilize Siderophore-Ferric Iron Uptake Transporter Systems for Activity against Gram-Negative Bacterial Pathogens.

Bryan EJ, Qiao Q, Wang Y, Roberge JY, LaVoie EJ, Pilch DS. Bryan EJ, et al. Among authors: roberge jy. Antibiotics (Basel). 2024 Feb 22;13(3):209. doi: 10.3390/antibiotics13030209. Antibiotics (Basel). 2024. PMID: 38534644 Free PMC article.

2

Structure-Activity Relationship of a Pyrrole Based Series of PfPKG Inhibitors as Anti-Malarials.

Gilleran JA, Ashraf K, Delvillar M, Eck T, Fondekar R, Miller EB, Hutchinson A, Dong A, Seitova A, De Souza ML, Augeri D, Halabelian L, Siekierka J, Rotella DP, Gordon J, Childers WE, Grier MC, Staker BL, Roberge JY, Bhanot P. Gilleran JA, et al. Among authors: roberge jy. J Med Chem. 2024 Mar 14;67(5):3467-3503. doi: 10.1021/acs.jmedchem.3c01795. Epub 2024 Feb 19. J Med Chem. 2024. PMID: 38372781

3

Structure-based design and optimization of a new class of small molecule inhibitors targeting the P-stalk binding pocket of ricin.

Rudolph MJ, Dutta A, Tsymbal AM, McLaughlin JE, Chen Y, Davis SA, Theodorous SA, Pierce M, Algava B, Zhang X, Szekely Z, Roberge JY, Li XP, Tumer NE. Rudolph MJ, et al. Among authors: roberge jy. Bioorg Med Chem. 2024 Feb 15;100:117614. doi: 10.1016/j.bmc.2024.117614. Epub 2024 Feb 5. Bioorg Med Chem. 2024. PMID: 38340640 Free article.

4

Acylpyrazoline-Based Third-Generation Selective Antichlamydial Compounds with Enhanced Potency.

Lu B, Qiao Q, Park ER, Wang Y, Gilleran JA, Pan M, Pilch DS, Wu X, Roberge JY, Fan H. Lu B, et al. Among authors: roberge jy. ACS Omega. 2023 Feb 8;8(7):6597-6607. doi: 10.1021/acsomega.2c06992. eCollection 2023 Feb 21. ACS Omega. 2023. PMID: 36844602 Free PMC article.

5

The Anticancer Drug Bleomycin Shows Potent Antifungal Activity by Altering Phospholipid Biosynthesis.

Pokharel M, Konarzewska P, Roberge JY, Han GS, Wang Y, Carman GM, Xue C. Pokharel M, et al. Among authors: roberge jy. Microbiol Spectr. 2022 Oct 26;10(5):e0086222. doi: 10.1128/spectrum.00862-22. Epub 2022 Aug 29. Microbiol Spectr. 2022. PMID: 36036637 Free PMC article.

6

TXH11106: A Third-Generation MreB Inhibitor with Enhanced Activity against a Broad Range of Gram-Negative Bacterial Pathogens.

Bryan EJ, Sagong HY, Parhi AK, Grier MC, Roberge JY, LaVoie EJ, Pilch DS. Bryan EJ, et al. Among authors: roberge jy. Antibiotics (Basel). 2022 May 20;11(5):693. doi: 10.3390/antibiotics11050693. Antibiotics (Basel). 2022. PMID: 35625337 Free PMC article.

7

Synthesis and Structural Characterization of Ricin Inhibitors Targeting Ribosome Binding Using Fragment-Based Methods and Structure-Based Design.

Li XP, Harijan RK, Cao B, Kahn JN, Pierce M, Tsymbal AM, Roberge JY, Augeri D, Tumer NE. Li XP, et al. Among authors: roberge jy. J Med Chem. 2021 Oct 28;64(20):15334-15348. doi: 10.1021/acs.jmedchem.1c01370. Epub 2021 Oct 14. J Med Chem. 2021. PMID: 34648707 Free PMC article.

8

A Novel Dual Drug Approach That Combines Ivermectin and Dihydromyricetin (DHM) to Reduce Alcohol Drinking and Preference in Mice.

Silva J, Carry E, Xue C, Zhang J, Liang J, Roberge JY, Davies DL. Silva J, et al. Among authors: roberge jy. Molecules. 2021 Mar 22;26(6):1791. doi: 10.3390/molecules26061791. Molecules. 2021. PMID: 33810134 Free PMC article.

9

Benzothiazolyl and Benzoxazolyl Hydrazones Function as Zinc Metallochaperones to Reactivate Mutant p53.

Gilleran JA, Yu X, Blayney AJ, Bencivenga AF, Na B, Augeri DJ, Blanden AR, Kimball SD, Loh SN, Roberge JY, Carpizo DR. Gilleran JA, et al. Among authors: roberge jy. J Med Chem. 2021 Feb 25;64(4):2024-2045. doi: 10.1021/acs.jmedchem.0c01360. Epub 2021 Feb 4. J Med Chem. 2021. PMID: 33538587 Free PMC article.

10

Design, synthesis, and biological evaluation of deuterated C-aryl glycoside as a potent and long-acting renal sodium-dependent glucose cotransporter 2 inhibitor for the treatment of type 2 diabetes.

Xu G, Lv B, Roberge JY, Xu B, Du J, Dong J, Chen Y, Peng K, Zhang L, Tang X, Feng Y, Xu M, Fu W, Zhang W, Zhu L, Deng Z, Sheng Z, Welihinda A, Sun X. Xu G, et al. Among authors: roberge jy. J Med Chem. 2014 Feb 27;57(4):1236-51. doi: 10.1021/jm401780b. Epub 2014 Feb 12. J Med Chem. 2014. PMID: 24456245

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