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New drug discovery strategies for the treatment of benznidazole-resistance in Trypanosoma cruzi, the causative agent of Chagas disease.
Expert Opin Drug Discov. 2024 May 7:1-13. doi: 10.1080/17460441.2024.2349155. Online ahead of print.
Expert Opin Drug Discov. 2024.
PMID: 38715393
Review.
Design and synthesis of benzofuran- and naphthalene-fused thiazinones as antimycobacterial agents.
Keiff F, Jacques Dit Lapierre TJW, Bernal FA, Kloss F.
Keiff F, et al. Among authors: jacques dit lapierre tjw.
Arch Pharm (Weinheim). 2023 Nov;356(11):e2300356. doi: 10.1002/ardp.202300356. Epub 2023 Sep 4.
Arch Pharm (Weinheim). 2023.
PMID: 37667452
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Hit-to-lead optimization of a pyrazinylpiperazine series against Leishmania infantum and Leishmania braziliensis.
Jacques Dit Lapierre TJW, Cruz MGFML, Brito NPF, Resende DM, Souza FO, Pilau EJ, da Silva MFB, Neves BJ, Murta SMF, Rezende Júnior CO.
Jacques Dit Lapierre TJW, et al.
Eur J Med Chem. 2023 Aug 5;256:115445. doi: 10.1016/j.ejmech.2023.115445. Epub 2023 May 2.
Eur J Med Chem. 2023.
PMID: 37156183
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