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Intrinsic thermodynamics of 4-substituted-2,3,5,6-tetrafluorobenzenesulfonamide binding to carbonic anhydrases by isothermal titration calorimetry.
Zubrienė A, Smirnovienė J, Smirnov A, Morkūnaitė V, Michailovienė V, Jachno J, Juozapaitienė V, Norvaišas P, Manakova E, Gražulis S, Matulis D. Zubrienė A, et al. Among authors: jachno j. Biophys Chem. 2015 Oct;205:51-65. doi: 10.1016/j.bpc.2015.05.009. Epub 2015 Jun 6. Biophys Chem. 2015. PMID: 26079542
Intrinsic thermodynamics of inhibitor binding to human carbonic anhydrase IX.
Linkuvienė V, Matulienė J, Juozapaitienė V, Michailovienė V, Jachno J, Matulis D. Linkuvienė V, et al. Among authors: jachno j. Biochim Biophys Acta. 2016 Apr;1860(4):708-18. doi: 10.1016/j.bbagen.2016.01.007. Epub 2016 Jan 18. Biochim Biophys Acta. 2016. PMID: 26794023
Intrinsic thermodynamics of high affinity inhibitor binding to recombinant human carbonic anhydrase IV.
Mickevičiūtė A, Timm DD, Gedgaudas M, Linkuvienė V, Chen Z, Waheed A, Michailovienė V, Zubrienė A, Smirnov A, Čapkauskaitė E, Baranauskienė L, Jachno J, Revuckienė J, Manakova E, Gražulis S, Matulienė J, Di Cera E, Sly WS, Matulis D. Mickevičiūtė A, et al. Among authors: jachno j. Eur Biophys J. 2018 Apr;47(3):271-290. doi: 10.1007/s00249-017-1256-0. Epub 2017 Oct 3. Eur Biophys J. 2018. PMID: 28975383 Free PMC article.
Inhibition and binding studies of carbonic anhydrase isozymes I, II and IX with benzimidazo[1,2-c][1,2,3]thiadiazole-7-sulphonamides.
Baranauskienė L, Hilvo M, Matulienė J, Golovenko D, Manakova E, Dudutienė V, Michailovienė V, Torresan J, Jachno J, Parkkila S, Maresca A, Supuran CT, Gražulis S, Matulis D. Baranauskienė L, et al. Among authors: jachno j. J Enzyme Inhib Med Chem. 2010 Dec;25(6):863-70. doi: 10.3109/14756360903571685. Epub 2010 Feb 18. J Enzyme Inhib Med Chem. 2010. PMID: 20166809
Discovery and characterization of novel selective inhibitors of carbonic anhydrase IX.
Dudutienė V, Matulienė J, Smirnov A, Timm DD, Zubrienė A, Baranauskienė L, Morkūnaite V, Smirnovienė J, Michailovienė V, Juozapaitienė V, Mickevičiūtė A, Kazokaitė J, Bakšytė S, Kasiliauskaitė A, Jachno J, Revuckienė J, Kišonaitė M, Pilipuitytė V, Ivanauskaitė E, Milinavičiūtė G, Smirnovas V, Petrikaitė V, Kairys V, Petrauskas V, Norvaišas P, Lingė D, Gibieža P, Capkauskaitė E, Zakšauskas A, Kazlauskas E, Manakova E, Gražulis S, Ladbury JE, Matulis D. Dudutienė V, et al. Among authors: jachno j. J Med Chem. 2014 Nov 26;57(22):9435-46. doi: 10.1021/jm501003k. Epub 2014 Nov 10. J Med Chem. 2014. PMID: 25358084
Picomolar fluorescent probes for compound affinity determination to carbonic anhydrase IX expressed in live cancer cells.
Matulienė J, Žvinys G, Petrauskas V, Kvietkauskaitė A, Zakšauskas A, Shubin K, Zubrienė A, Baranauskienė L, Kačenauskaitė L, Kopanchuk S, Veiksina S, Paketurytė-Latvė V, Smirnovienė J, Juozapaitienė V, Mickevičiūtė A, Michailovienė V, Jachno J, Stravinskienė D, Sližienė A, Petrošiūtė A, Becker HM, Kazokaitė-Adomaitienė J, Yaromina A, Čapkauskaitė E, Rinken A, Dudutienė V, Dubois LJ, Matulis D. Matulienė J, et al. Among authors: jachno j. Sci Rep. 2022 Oct 21;12(1):17644. doi: 10.1038/s41598-022-22436-1. Sci Rep. 2022. PMID: 36271018 Free PMC article.
14 results