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Table representation of search results timeline featuring number of search results per year.

Year Number of Results
2003 1
2004 1
2005 8
2006 7
2007 6
2008 8
2009 9
2010 12
2011 18
2012 16
2013 10
2014 5
2015 8
2016 5
2017 2
2018 8
2019 12
2020 7
2021 9
2022 6
2023 9
2024 4

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152 results

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Page 1
Pharmacological Characterization and Radiolabeling of VUF15485, a High-Affinity Small-Molecule Agonist for the Atypical Chemokine Receptor ACKR3.
Zarca AM, Adlere I, Viciano CP, Arimont-Segura M, Meyrath M, Simon IA, Bebelman JP, Laan D, Custers HGJ, Janssen E, Versteegh KL, Buzink MCML, Nesheva DN, Bosma R, de Esch IJP, Vischer HF, Wijtmans M, Szpakowska M, Chevigné A, Hoffmann C, de Graaf C, Zarzycka BA, Windhorst AD, Smit MJ, Leurs R. Zarca AM, et al. Among authors: de esch ijp. Mol Pharmacol. 2024 Mar 14;105(4):301-312. doi: 10.1124/molpharm.123.000835. Mol Pharmacol. 2024. PMID: 38346795
Fragment-to-Lead Medicinal Chemistry Publications in 2022.
Woodhead AJ, Erlanson DA, de Esch IJP, Holvey RS, Jahnke W, Pathuri P. Woodhead AJ, et al. Among authors: de esch ijp. J Med Chem. 2024 Feb 22;67(4):2287-2304. doi: 10.1021/acs.jmedchem.3c02070. Epub 2024 Jan 30. J Med Chem. 2024. PMID: 38289623 Review.
Multiplexed experimental strategies for fragment library screening against challenging drug targets using SPR biosensors.
FitzGerald EA, Vagrys D, Opassi G, Klein HF, Hamilton DJ, Talibov VO, Abramsson M, Moberg A, Lindgren MT, Holmgren C, Davis B, O'Brien P, Wijtmans M, Hubbard RE, de Esch IJP, Danielson UH. FitzGerald EA, et al. Among authors: de esch ijp. SLAS Discov. 2024 Jan;29(1):40-51. doi: 10.1016/j.slasd.2023.09.001. Epub 2023 Sep 14. SLAS Discov. 2024. PMID: 37714432 Free article.
An Automated, Open-Source Workflow for the Generation of (3D) Fragment Libraries.
Dekker T, Janssen MACH, Sutherland C, Aben RWM, Scheeren HW, Blanco-Ania D, Rutjes FPJT, Wijtmans M, de Esch IJP. Dekker T, et al. Among authors: de esch ijp. ACS Med Chem Lett. 2023 May 2;14(5):583-590. doi: 10.1021/acsmedchemlett.2c00503. eCollection 2023 May 11. ACS Med Chem Lett. 2023. PMID: 37197454 Free PMC article.
To Target or Not to Target Schistosoma mansoni Cyclic Nucleotide Phosphodiesterase 4A?
Zheng Y, Schroeder S, Kanev GK, Botros SS, William S, Sabra AA, Maes L, Caljon G, Gil C, Martinez A, Salado IG, Augustyns K, Edink E, Sijm M, de Heuvel E, de Esch IJP, van der Meer T, Siderius M, Sterk GJ, Brown D, Leurs R. Zheng Y, et al. Among authors: de esch ijp. Int J Mol Sci. 2023 Apr 6;24(7):6817. doi: 10.3390/ijms24076817. Int J Mol Sci. 2023. PMID: 37047792 Free PMC article.
152 results