Inoue A - Search Results

1

Design and Characterization of an Intracellular Covalent Ligand for CC Chemokine Receptor 2.

Ortiz Zacarías NV, Chahal KK, Šimková T, van der Horst C, Zheng Y, Inoue A, Theunissen E, Mallee L, van der Es D, Louvel J, IJzerman AP, Handel TM, Kufareva I, Heitman LH. Ortiz Zacarías NV, et al. Among authors: inoue a. J Med Chem. 2021 Mar 11;64(5):2608-2621. doi: 10.1021/acs.jmedchem.0c01137. Epub 2021 Feb 18. J Med Chem. 2021. PMID: 33600174 Free PMC article.

2

Synthesis and biological evaluation of optically active Ki16425.

Sato T, Sugimoto K, Inoue A, Okudaira S, Aoki J, Tokuyama H. Sato T, et al. Among authors: inoue a. Bioorg Med Chem Lett. 2012 Jul 1;22(13):4323-6. doi: 10.1016/j.bmcl.2012.05.012. Epub 2012 May 11. Bioorg Med Chem Lett. 2012. PMID: 22658556

3

Conformational Constraint of the Glycerol Moiety of Lysophosphatidylserine Affords Compounds with Receptor Subtype Selectivity.

Jung S, Inoue A, Nakamura S, Kishi T, Uwamizu A, Sayama M, Ikubo M, Otani Y, Kano K, Makide K, Aoki J, Ohwada T. Jung S, et al. Among authors: inoue a. J Med Chem. 2016 Apr 28;59(8):3750-76. doi: 10.1021/acs.jmedchem.5b01925. Epub 2016 Apr 14. J Med Chem. 2016. PMID: 27077565

4

Probing the Hydrophobic Binding Pocket of G-Protein-Coupled Lysophosphatidylserine Receptor GPR34/LPS₁ by Docking-Aided Structure-Activity Analysis.

Sayama M, Inoue A, Nakamura S, Jung S, Ikubo M, Otani Y, Uwamizu A, Kishi T, Makide K, Aoki J, Hirokawa T, Ohwada T. Sayama M, et al. Among authors: inoue a. J Med Chem. 2017 Jul 27;60(14):6384-6399. doi: 10.1021/acs.jmedchem.7b00693. Epub 2017 Jul 17. J Med Chem. 2017. PMID: 28715213

5

Non-naturally Occurring Regio Isomer of Lysophosphatidylserine Exhibits Potent Agonistic Activity toward G Protein-Coupled Receptors.

Nakamura S, Sayama M, Uwamizu A, Jung S, Ikubo M, Otani Y, Kano K, Omi J, Inoue A, Aoki J, Ohwada T. Nakamura S, et al. Among authors: inoue a. J Med Chem. 2020 Sep 10;63(17):9990-10029. doi: 10.1021/acs.jmedchem.0c01126. Epub 2020 Aug 24. J Med Chem. 2020. PMID: 32787112

6

Switching Lysophosphatidylserine G Protein-Coupled Receptor Agonists to Antagonists by Acylation of the Hydrophilic Serine Amine.

Sayama M, Uwamizu A, Ikubo M, Chen L, Yan G, Otani Y, Inoue A, Aoki J, Ohwada T. Sayama M, et al. Among authors: inoue a. J Med Chem. 2021 Jul 22;64(14):10059-10101. doi: 10.1021/acs.jmedchem.1c00347. Epub 2021 Jul 7. J Med Chem. 2021. PMID: 34233115

7

Synthesis of unnatural morphinan compounds to induce itch-like behaviors in mice: Towards the development of MRGPRX2 selective ligands.

Iio K, Kutsumura N, Nagumo Y, Saitoh T, Tokuda A, Hashimoto K, Yamamoto N, Kise R, Inoue A, Mizoguchi H, Nagase H. Iio K, et al. Among authors: inoue a. Bioorg Med Chem Lett. 2022 Jan 15;56:128485. doi: 10.1016/j.bmcl.2021.128485. Epub 2021 Nov 30. Bioorg Med Chem Lett. 2022. PMID: 34861349

8

Exploration of LPS₂ agonist binding modes using the combination of a new hydrophobic scaffold and homology modeling.

Chen L, Uwamizu A, Sayama M, Kano K, Otani Y, Kondo S, Inoue A, Aoki J, Ohwada T. Chen L, et al. Among authors: inoue a. Eur J Med Chem. 2023 Apr 5;252:115271. doi: 10.1016/j.ejmech.2023.115271. Epub 2023 Mar 11. Eur J Med Chem. 2023. PMID: 36965226

9

Design and Synthesis of Orexin 1 Receptor-Selective Agonists.

Iio K, Hashimoto K, Nagumo Y, Amezawa M, Hasegawa T, Yamamoto N, Kutsumura N, Takeuchi K, Ishikawa Y, Yamamoto H, Tokuda A, Sato T, Uchida Y, Inoue A, Tanimura R, Yanagisawa M, Nagase H, Saitoh T. Iio K, et al. Among authors: inoue a. J Med Chem. 2023 Apr 27;66(8):5453-5464. doi: 10.1021/acs.jmedchem.2c01773. Epub 2023 Apr 12. J Med Chem. 2023. PMID: 37043436

10

Phosphorothioate analogs of sn-2 radyl lysophosphatidic acid (LPA): metabolically stabilized LPA receptor agonists.

Jiang G, Inoue A, Aoki J, Prestwich GD. Jiang G, et al. Among authors: inoue a. Bioorg Med Chem Lett. 2013 Mar 15;23(6):1865-9. doi: 10.1016/j.bmcl.2013.01.002. Epub 2013 Jan 23. Bioorg Med Chem Lett. 2013. PMID: 23395664

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