Poor and enantioselective bioavailability of naftopidil enantiomers is due to extensive and stereoselective metabolism in rat liver.
Liu X, Zhu L, Huang B, Huang J, Cai Y, Zhu L, Wu B, Fu X, Zhang X, Rong Y, Xiao Q, Guo J, Li A, Guo Y, Yuan M.
Liu X, et al. Among authors: huang b, huang j.
J Pharm Biomed Anal. 2017 Jan 5;132:165-172. doi: 10.1016/j.jpba.2016.09.038. Epub 2016 Sep 27.
J Pharm Biomed Anal. 2017.
PMID: 27744175