Structure-activity relationship for the folding intermediate-selective inhibition of DYRK1A.
Miyazaki Y, Kikuchi M, Umezawa K, Descamps A, Nakamura D, Furuie G, Sumida T, Saito K, Kimura N, Niwa T, Sumida Y, Umehara T, Hosoya T, Kii I.
Miyazaki Y, et al. Among authors: hosoya t.
Eur J Med Chem. 2022 Jan 5;227:113948. doi: 10.1016/j.ejmech.2021.113948. Epub 2021 Oct 28.
Eur J Med Chem. 2022.
PMID: 34742017