Heinrich MR - Search Results

1

Selectfluor-Mediated Chlorination and Fluorination of Arenes: Late-Stage Functionalization of APIs and Its Biological Effects.

Gradl S, Zantop V, Gmeiner P, Hübner H, Heinrich MR. Gradl S, et al. Among authors: heinrich mr. ChemMedChem. 2023 Aug 1;18(15):e202300144. doi: 10.1002/cmdc.202300144. Epub 2023 May 8. ChemMedChem. 2023. PMID: 37088715

2

Synthesis, biological evaluation and radiolabelling by 18F-fluoroarylation of a dopamine D3-selective ligand as prospective imaging probe for PET.

Höfling SB, Maschauer S, Hübner H, Gmeiner P, Wester HJ, Prante O, Heinrich MR. Höfling SB, et al. Among authors: heinrich mr. Bioorg Med Chem Lett. 2010 Dec 1;20(23):6933-7. doi: 10.1016/j.bmcl.2010.09.142. Epub 2010 Oct 26. Bioorg Med Chem Lett. 2010. PMID: 21030255

3

Radical arylation of tyrosine and its application in the synthesis of a highly selective neurotensin receptor 2 ligand.

Pratsch G, Unfried JF, Einsiedel J, Plomer M, Hübner H, Gmeiner P, Heinrich MR. Pratsch G, et al. Among authors: heinrich mr. Org Biomol Chem. 2011 May 21;9(10):3746-52. doi: 10.1039/c1ob05292f. Epub 2011 Apr 6. Org Biomol Chem. 2011. PMID: 21472182

4

Fast and efficient (18) F-labeling by [(18) f]fluorophenylazocarboxylic esters.

Fehler SK, Maschauer S, Höfling SB, Bartuschat AL, Tschammer N, Hübner H, Gmeiner P, Prante O, Heinrich MR. Fehler SK, et al. Among authors: heinrich mr. Chemistry. 2014 Jan 7;20(2):370-5. doi: 10.1002/chem.201303409. Epub 2013 Dec 11. Chemistry. 2014. PMID: 24339325

5

Synthesis and evaluation of fluoro substituted pyridinylcarboxamides and their phenylazo analogues for potential dopamine D3 receptor PET imaging.

Nebel N, Maschauer S, Bartuschat AL, Fehler SK, Hübner H, Gmeiner P, Kuwert T, Heinrich MR, Prante O, Hocke C. Nebel N, et al. Among authors: heinrich mr. Bioorg Med Chem Lett. 2014 Dec 1;24(23):5399-403. doi: 10.1016/j.bmcl.2014.10.043. Bioorg Med Chem Lett. 2014. PMID: 25453796

6

Fluoro-substituted phenylazocarboxamides: Dopaminergic behavior and N-arylating properties for irreversible binding.

Bartuschat AL, Schellhorn T, Hübner H, Gmeiner P, Heinrich MR. Bartuschat AL, et al. Among authors: heinrich mr. Bioorg Med Chem. 2015 Jul 15;23(14):3938-47. doi: 10.1016/j.bmc.2014.12.012. Epub 2014 Dec 17. Bioorg Med Chem. 2015. PMID: 25564378

7

[¹⁸F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor.

Nebel N, Strauch B, Maschauer S, Lasch R, Rampp H, Fehler SK, Bock LR, Hübner H, Gmeiner P, Heinrich MR, Prante O. Nebel N, et al. Among authors: heinrich mr. ACS Omega. 2017 Dec 31;2(12):8649-8659. doi: 10.1021/acsomega.7b01374. Epub 2017 Dec 6. ACS Omega. 2017. PMID: 29479577 Free PMC article.

8

Structure-guided development of selective M3 muscarinic acetylcholine receptor antagonists.

Liu H, Hofmann J, Fish I, Schaake B, Eitel K, Bartuschat A, Kaindl J, Rampp H, Banerjee A, Hübner H, Clark MJ, Vincent SG, Fisher JT, Heinrich MR, Hirata K, Liu X, Sunahara RK, Shoichet BK, Kobilka BK, Gmeiner P. Liu H, et al. Among authors: heinrich mr. Proc Natl Acad Sci U S A. 2018 Nov 20;115(47):12046-12050. doi: 10.1073/pnas.1813988115. Epub 2018 Nov 7. Proc Natl Acad Sci U S A. 2018. PMID: 30404914 Free PMC article.

9

Benzyl Phenylsemicarbazides: A Chemistry-Driven Approach Leading to G Protein-Biased Dopamine D₄ Receptor Agonists with High Subtype Selectivity.

Pirzer AS, Lasch R, Friedrich H, Hübner H, Gmeiner P, Heinrich MR. Pirzer AS, et al. Among authors: heinrich mr. J Med Chem. 2019 Nov 14;62(21):9658-9679. doi: 10.1021/acs.jmedchem.9b01085. Epub 2019 Oct 30. J Med Chem. 2019. PMID: 31613617

10

Aryl Radical Selectivity in Biphasic Systems.

Altmann LM, Fürst MCD, Gans EI, Zantop V, Pratsch G, Heinrich MR. Altmann LM, et al. Among authors: heinrich mr. Org Lett. 2020 Jan 17;22(2):479-482. doi: 10.1021/acs.orglett.9b04237. Epub 2020 Jan 6. Org Lett. 2020. PMID: 31904970

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