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Targeting metabolic activity in high-risk neuroblastoma through Monocarboxylate Transporter 1 (MCT1) inhibition.
Oncogene. 2020 Apr;39(17):3555-3570. doi: 10.1038/s41388-020-1235-2. Epub 2020 Mar 2.
Oncogene. 2020.
PMID: 32123312
Free PMC article.
Suppression of the ATP-binding cassette transporter ABCC4 impairs neuroblastoma tumour growth and sensitises to irinotecan in vivo.
Murray J, Valli E, Yu DMT, Truong AM, Gifford AJ, Eden GL, Gamble LD, Hanssen KM, Flemming CL, Tan A, Tivnan A, Allan S, Saletta F, Cheung L, Ruhle M, Schuetz JD, Henderson MJ, Byrne JA, Norris MD, Haber M, Fletcher JI.
Murray J, et al. Among authors: hanssen km.
Eur J Cancer. 2017 Sep;83:132-141. doi: 10.1016/j.ejca.2017.06.024. Epub 2017 Jul 20.
Eur J Cancer. 2017.
PMID: 28735070
Free PMC article.
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Inhibition of polyamine synthesis and uptake reduces tumor progression and prolongs survival in mouse models of neuroblastoma.
Gamble LD, Purgato S, Murray J, Xiao L, Yu DMT, Hanssen KM, Giorgi FM, Carter DR, Gifford AJ, Valli E, Milazzo G, Kamili A, Mayoh C, Liu B, Eden G, Sarraf S, Allan S, Di Giacomo S, Flemming CL, Russell AJ, Cheung BB, Oberthuer A, London WB, Fischer M, Trahair TN, Fletcher JI, Marshall GM, Ziegler DS, Hogarty MD, Burns MR, Perini G, Norris MD, Haber M.
Gamble LD, et al. Among authors: hanssen km.
Sci Transl Med. 2019 Jan 30;11(477):eaau1099. doi: 10.1126/scitranslmed.aau1099.
Sci Transl Med. 2019.
PMID: 30700572
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MRP1 modulators synergize with buthionine sulfoximine to exploit collateral sensitivity and selectively kill MRP1-expressing cancer cells.
Gana CC, Hanssen KM, Yu DMT, Flemming CL, Wheatley MS, Conseil G, Cole SPC, Norris MD, Haber M, Fletcher JI.
Gana CC, et al. Among authors: hanssen km.
Biochem Pharmacol. 2019 Oct;168:237-248. doi: 10.1016/j.bcp.2019.07.009. Epub 2019 Jul 11.
Biochem Pharmacol. 2019.
PMID: 31302132
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Targeting multidrug resistance-associated protein 1 (MRP1)-expressing cancers: Beyond pharmacological inhibition.
Hanssen KM, Haber M, Fletcher JI.
Hanssen KM, et al.
Drug Resist Updat. 2021 Dec;59:100795. doi: 10.1016/j.drup.2021.100795. Epub 2021 Dec 10.
Drug Resist Updat. 2021.
PMID: 34983733
Review.
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GSH facilitates the binding and inhibitory activity of novel multidrug resistance protein 1 (MRP1) modulators.
Hanssen KM, Wheatley MS, Yu DMT, Conseil G, Norris MD, Haber M, Cole SPC, Fletcher JI.
Hanssen KM, et al.
FEBS J. 2022 Jul;289(13):3854-3875. doi: 10.1111/febs.16374. Epub 2022 Feb 8.
FEBS J. 2022.
PMID: 35080351
Free article.
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Generation of Orthotopic and Subcutaneous Patient-Derived Xenograft Models from Diverse Clinical Tissue Samples of Pediatric Extracranial Solid Tumors.
Hanssen KM, Fletcher JI, Kamili A.
Hanssen KM, et al.
Methods Mol Biol. 2024;2806:55-74. doi: 10.1007/978-1-0716-3858-3_6.
Methods Mol Biol. 2024.
PMID: 38676796
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