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Development of novel cyclic peptides as pro-apoptotic agents.
Brindisi M, Maramai S, Brogi S, Fanigliulo E, Butini S, Guarino E, Casagni A, Lamponi S, Bonechi C, Nathwani SM, Finetti F, Ragonese F, Arcidiacono P, Campiglia P, Valenti S, Novellino E, Spaccapelo R, Morbidelli L, Zisterer DM, Williams CD, Donati A, Baldari C, Campiani G, Ulivieri C, Gemma S. Brindisi M, et al. Among authors: guarino e. Eur J Med Chem. 2016 Jul 19;117:301-20. doi: 10.1016/j.ejmech.2016.04.001. Epub 2016 Apr 5. Eur J Med Chem. 2016. PMID: 27150036
1H-cyclopentapyrimidine-2,4(1H,3H)-dione-related ionotropic glutamate receptors ligands. structure-activity relationships and identification of potent and Selective iGluR5 modulators.
Butini S, Pickering DS, Morelli E, Coccone SS, Trotta F, De Angelis M, Guarino E, Fiorini I, Campiani G, Novellino E, Schousboe A, Christensen JK, Gemma S. Butini S, et al. Among authors: guarino e. J Med Chem. 2008 Oct 23;51(20):6614-8. doi: 10.1021/jm800865a. Epub 2008 Sep 24. J Med Chem. 2008. PMID: 18811139
A stereoselective approach to peptidomimetic BACE1 inhibitors.
Butini S, Gabellieri E, Brindisi M, Giovani S, Maramai S, Kshirsagar G, Guarino E, Brogi S, La Pietra V, Giustiniano M, Marinelli L, Novellino E, Campiani G, Cappelli A, Gemma S. Butini S, et al. Among authors: guarino e. Eur J Med Chem. 2013;70:233-47. doi: 10.1016/j.ejmech.2013.09.056. Epub 2013 Oct 6. Eur J Med Chem. 2013. PMID: 24158015
Discovery of bishomo(hetero)arylpiperazines as novel multifunctional ligands targeting dopamine D(3) and serotonin 5-HT(1A) and 5-HT(2A) receptors.
Butini S, Campiani G, Franceschini S, Trotta F, Kumar V, Guarino E, Borrelli G, Fiorini I, Novellino E, Fattorusso C, Persico M, Orteca N, Sandager-Nielsen K, Jacobsen TA, Madsen K, Scheel-Kruger J, Gemma S. Butini S, et al. Among authors: guarino e. J Med Chem. 2010 Jun 24;53(12):4803-7. doi: 10.1021/jm100294b. J Med Chem. 2010. PMID: 20481570
Selective kainate receptor (GluK1) ligands structurally based upon 1H-cyclopentapyrimidin-2,4(1H,3H)-dione: synthesis, molecular modeling, and pharmacological and biostructural characterization.
Venskutonyte R, Butini S, Coccone SS, Gemma S, Brindisi M, Kumar V, Guarino E, Maramai S, Valenti S, Amir A, Valadés EA, Frydenvang K, Kastrup JS, Novellino E, Campiani G, Pickering DS. Venskutonyte R, et al. Among authors: guarino e. J Med Chem. 2011 Jul 14;54(13):4793-805. doi: 10.1021/jm2004078. Epub 2011 Jun 13. J Med Chem. 2011. PMID: 21619066
Multifunctional cholinesterase and amyloid Beta fibrillization modulators. Synthesis and biological investigation.
Butini S, Brindisi M, Brogi S, Maramai S, Guarino E, Panico A, Saxena A, Chauhan V, Colombo R, Verga L, De Lorenzi E, Bartolini M, Andrisano V, Novellino E, Campiani G, Gemma S. Butini S, et al. Among authors: guarino e. ACS Med Chem Lett. 2013 Oct 6;4(12):1178-82. doi: 10.1021/ml4002908. eCollection 2013 Dec 12. ACS Med Chem Lett. 2013. PMID: 24900626 Free PMC article.
88 results