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Boronic acid inhibitors of penicillin-binding protein 1b: serine and lysine labelling agents.
J Enzyme Inhib Med Chem. 2024 Dec;39(1):2305833. doi: 10.1080/14756366.2024.2305833. Epub 2024 Feb 27.
J Enzyme Inhib Med Chem. 2024.
PMID: 38410950
Free PMC article.
Next-Generation Heterocyclic Electrophiles as Small-Molecule Covalent MurA Inhibitors.
Ábrányi-Balogh P, Keeley A, Ferenczy GG, Petri L, Imre T, Grabrijan K, Hrast M, Knez D, Ilaš J, Gobec S, Keserű GM.
Ábrányi-Balogh P, et al. Among authors: grabrijan k.
Pharmaceuticals (Basel). 2022 Nov 29;15(12):1484. doi: 10.3390/ph15121484.
Pharmaceuticals (Basel). 2022.
PMID: 36558935
Free PMC article.
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Fragment-Sized Thiazoles in Fragment-Based Drug Discovery Campaigns: Friend or Foe?
Proj M, Hrast M, Knez D, Bozovičar K, Grabrijan K, Meden A, Gobec S, Frlan R.
Proj M, et al. Among authors: grabrijan k.
ACS Med Chem Lett. 2022 Nov 3;13(12):1905-1910. doi: 10.1021/acsmedchemlett.2c00429. eCollection 2022 Dec 8.
ACS Med Chem Lett. 2022.
PMID: 36518695
Free PMC article.
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Covalent inhibitors of bacterial peptidoglycan biosynthesis enzyme MurA with chloroacetamide warhead.
Grabrijan K, Hrast M, Proj M, Dolšak A, Zdovc I, Imre T, Petri L, Ábrányi-Balogh P, Keserű GM, Gobec S.
Grabrijan K, et al.
Eur J Med Chem. 2022 Dec 5;243:114752. doi: 10.1016/j.ejmech.2022.114752. Epub 2022 Sep 13.
Eur J Med Chem. 2022.
PMID: 36126388
Free article.
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Synthesis of 3-Amino-4-substituted Monocyclic ß-Lactams-Important Structural Motifs in Medicinal Chemistry.
Grabrijan K, Strašek N, Gobec S.
Grabrijan K, et al.
Int J Mol Sci. 2021 Dec 29;23(1):360. doi: 10.3390/ijms23010360.
Int J Mol Sci. 2021.
PMID: 35008788
Free PMC article.
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Design, synthesis and biological evaluation of substituted 3-amino-N-(thiazol-2-yl)pyrazine-2-carboxamides as inhibitors of mycobacterial methionine aminopeptidase 1.
Juhás M, Pallabothula VSK, Grabrijan K, Šimovičová M, Janďourek O, Konečná K, Bárta P, Paterová P, Gobec S, Sosič I, Zitko J.
Juhás M, et al. Among authors: grabrijan k.
Bioorg Chem. 2022 Jan;118:105489. doi: 10.1016/j.bioorg.2021.105489. Epub 2021 Nov 14.
Bioorg Chem. 2022.
PMID: 34826708
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Monocyclic beta-lactams for therapeutic uses: a patent overview (2010-2020).
Grabrijan K, Strašek N, Gobec S.
Grabrijan K, et al.
Expert Opin Ther Pat. 2021 Mar;31(3):247-266. doi: 10.1080/13543776.2021.1865919. Epub 2021 Jan 7.
Expert Opin Ther Pat. 2021.
PMID: 33327805
Review.
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Chlorocarbonylsulfenyl Chloride Cyclizations Towards Piperidin-3-yl-oxathiazol-2-ones as Potential Covalent Inhibitors of Threonine Proteases.
Jukič M, Grabrijan K, Kadić S, Lera Garrido FJ, Sosič I, Gobec S, Obreza A.
Jukič M, et al. Among authors: grabrijan k.
Acta Chim Slov. 2017 Dec;64(4):771-781. doi: 10.17344/acsi.2017.3883.
Acta Chim Slov. 2017.
PMID: 29318298
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