Glawar AF - Search Results

1

Nine of 16 stereoisomeric polyhydroxylated proline amides are potent β-N-acetylhexosaminidase inhibitors.

Ayers BJ, Glawar AF, Martínez RF, Ngo N, Liu Z, Fleet GW, Butters TD, Nash RJ, Yu CY, Wormald MR, Nakagawa S, Adachi I, Kato A, Jenkinson SF. Ayers BJ, et al. Among authors: glawar af. J Org Chem. 2014 Apr 18;79(8):3398-409. doi: 10.1021/jo500157p. Epub 2014 Apr 7. J Org Chem. 2014. PMID: 24641544

2

Structural essentials for β-N-acetylhexosaminidase inhibition by amides of prolines, pipecolic and azetidine carboxylic acids.

Glawar AF, Martínez RF, Ayers BJ, Hollas MA, Ngo N, Nakagawa S, Kato A, Butters TD, Fleet GW, Jenkinson SF. Glawar AF, et al. Org Biomol Chem. 2016 Nov 8;14(44):10371-10385. doi: 10.1039/c6ob01549b. Org Biomol Chem. 2016. PMID: 27735004

3

Synthesis from D-altrose of (5R,6R,7R,8S)-5,7-dihydroxy-8-hydroxymethylconidine and 2,4-dideoxy-2,4-imino-D-glucitol, azetidine analogues of swainsonine and 1,4-dideoxy-1,4-imino-D-mannitol.

Araújo N, Jenkinson SF, Martínez RF, Glawar AF, Wormald MR, Butters TD, Nakagawa S, Adachi I, Kato A, Yoshihara A, Akimitsu K, Izumori K, Fleet GW. Araújo N, et al. Among authors: glawar af. Org Lett. 2012 Aug 17;14(16):4174-7. doi: 10.1021/ol301844n. Epub 2012 Jul 27. Org Lett. 2012. PMID: 22839435

4

3-Hydroxyazetidine carboxylic acids: non-proteinogenic amino acids for medicinal chemists.

Glawar AF, Jenkinson SF, Thompson AL, Nakagawa S, Kato A, Butters TD, Fleet GW. Glawar AF, et al. ChemMedChem. 2013 Apr;8(4):658-66. doi: 10.1002/cmdc.201200541. Epub 2013 Mar 6. ChemMedChem. 2013. PMID: 23468173

5

An approach to 8 stereoisomers of homonojirimycin from (D)-glucose via kinetic & thermodynamic azido-γ-lactones.

Glawar AF, Jenkinson SF, Newberry SJ, Thompson AL, Nakagawa S, Yoshihara A, Akimitsu K, Izumori K, Butters TD, Kato A, Fleet GW. Glawar AF, et al. Org Biomol Chem. 2013 Sep 25;11(40):6886-99. doi: 10.1039/c3ob41334a. Org Biomol Chem. 2013. PMID: 23963282

6

Synthesis of the enantiomers of XYLNAc and LYXNAc: comparison of β-N-acetylhexosaminidase inhibition by the 8 stereoisomers of 2-N-acetylamino-1,2,4-trideoxy-1,4-iminopentitols.

Crabtree EV, Martínez RF, Nakagawa S, Adachi I, Butters TD, Kato A, Fleet GW, Glawar AF. Crabtree EV, et al. Among authors: glawar af. Org Biomol Chem. 2014 Jun 21;12(23):3932-43. doi: 10.1039/c4ob00097h. Org Biomol Chem. 2014. PMID: 24802185

7

Scalable syntheses of both enantiomers of DNJNAc and DGJNAc from glucuronolactone: the effect of N-alkylation on hexosaminidase inhibition.

Glawar AF, Best D, Ayers BJ, Miyauchi S, Nakagawa S, Aguilar-Moncayo M, García Fernández JM, Ortiz Mellet C, Crabtree EV, Butters TD, Wilson FX, Kato A, Fleet GW. Glawar AF, et al. Chemistry. 2012 Jul 23;18(30):9341-59. doi: 10.1002/chem.201200110. Epub 2012 Jun 26. Chemistry. 2012. PMID: 22736508

8

Short and sweet: (D)-glucose to (L)-glucose and (L)-glucuronic acid.

Martínez RF, Liu Z, Glawar AF, Yoshihara A, Izumori K, Fleet GW, Jenkinson SF. Martínez RF, et al. Among authors: glawar af. Angew Chem Int Ed Engl. 2014 Jan 20;53(4):1160-2. doi: 10.1002/anie.201309073. Epub 2013 Dec 5. Angew Chem Int Ed Engl. 2014. PMID: 24310928

9

2-Acetamido-N-benzyl-1,4-imino-1,2,4-tride-oxy-l-xylitol (N-benzyl-l-XYLNAc).

Jenkinson SF, Crabtree EV, Glawar AF, Butters TD, Fleet GW, Watkin DJ. Jenkinson SF, et al. Among authors: glawar af. Acta Crystallogr Sect E Struct Rep Online. 2010 Apr 24;66(Pt 5):o1147-8. doi: 10.1107/S1600536810014145. Acta Crystallogr Sect E Struct Rep Online. 2010. PMID: 21579195 Free PMC article.

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