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Page 1
Synthesis and structure-activity relationship studies in translocator protein ligands based on a pyrazolo[3,4-b]quinoline scaffold.
Cappelli A, Bini G, Valenti S, Giuliani G, Paolino M, Anzini M, Vomero S, Giorgi G, Giordani A, Stasi LP, Makovec F, Ghelardini C, Di Cesare Mannelli L, Concas A, Porcu P, Biggio G. Cappelli A, et al. Among authors: giordani a. J Med Chem. 2011 Oct 27;54(20):7165-75. doi: 10.1021/jm200770f. Epub 2011 Sep 26. J Med Chem. 2011. PMID: 21916402
Design, synthesis, and biological evaluation of AT1 angiotensin II receptor antagonists based on the pyrazolo[3,4-b]pyridine and related heteroaromatic bicyclic systems.
Cappelli A, Nannicini C, Gallelli A, Giuliani G, Valenti S, Mohr Gl, Anzini M, Mennuni L, Ferrari F, Caselli G, Giordani A, Peris W, Makovec F, Giorgi G, Vomero S. Cappelli A, et al. Among authors: giordani a. J Med Chem. 2008 Apr 10;51(7):2137-46. doi: 10.1021/jm7011563. Epub 2008 Mar 5. J Med Chem. 2008. PMID: 18318468
Progress towards the identification of new aggrecanase inhibitors.
De Rienzo F, Saxena P, Filomia F, Caselli G, Colace F, Stasi L, Giordani A, Menziani MC. De Rienzo F, et al. Among authors: giordani a. Curr Med Chem. 2009;16(19):2395-415. doi: 10.2174/092986709788682092. Curr Med Chem. 2009. PMID: 19601788 Review.
Synthesis and biological evaluation of amidine, guanidine, and thiourea derivatives of 2-amino(6-trifluoromethoxy)benzothiazole as neuroprotective agents potentially useful in brain diseases.
Anzini M, Chelini A, Mancini A, Cappelli A, Frosini M, Ricci L, Valoti M, Magistretti J, Castelli L, Giordani A, Makovec F, Vomero S. Anzini M, et al. Among authors: giordani a. J Med Chem. 2010 Jan 28;53(2):734-44. doi: 10.1021/jm901375r. J Med Chem. 2010. PMID: 19950903
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
Cappelli A, Manini M, Valenti S, Castriconi F, Giuliani G, Anzini M, Brogi S, Butini S, Gemma S, Campiani G, Giorgi G, Mennuni L, Lanza M, Giordani A, Caselli G, Letari O, Makovec F. Cappelli A, et al. Among authors: giordani a. Eur J Med Chem. 2013 May;63:85-94. doi: 10.1016/j.ejmech.2013.01.044. Epub 2013 Feb 8. Eur J Med Chem. 2013. PMID: 23466604
Novel analgesic/anti-inflammatory agents: 1,5-diarylpyrrole nitrooxyalkyl ethers and related compounds as cyclooxygenase-2 inhibiting nitric oxide donors.
Anzini M, Di Capua A, Valenti S, Brogi S, Rovini M, Giuliani G, Cappelli A, Vomero S, Chiasserini L, Sega A, Poce G, Giorgi G, Calderone V, Martelli A, Testai L, Sautebin L, Rossi A, Pace S, Ghelardini C, Di Cesare Mannelli L, Benetti V, Giordani A, Anzellotti P, Dovizio M, Patrignani P, Biava M. Anzini M, et al. Among authors: giordani a. J Med Chem. 2013 Apr 25;56(8):3191-206. doi: 10.1021/jm301370e. Epub 2013 Apr 11. J Med Chem. 2013. PMID: 23534442
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity.
Di Capua A, Sticozzi C, Brogi S, Brindisi M, Cappelli A, Sautebin L, Rossi A, Pace S, Ghelardini C, Di Cesare Mannelli L, Valacchi G, Giorgi G, Giordani A, Poce G, Biava M, Anzini M. Di Capua A, et al. Among authors: giordani a. Eur J Med Chem. 2016 Feb 15;109:99-106. doi: 10.1016/j.ejmech.2015.12.044. Epub 2015 Dec 28. Eur J Med Chem. 2016. PMID: 26774035
Phenylindenone isomers as divergent modulators of p38α MAP kinase.
Cappelli A, Nannicini C, Chelini A, Paolino M, Giuliani G, Anzini M, Giordani A, Sabatini C, Caselli G, Mennuni L, Makovec F, Giorgi G, Vomero S, Menziani MC. Cappelli A, et al. Among authors: giordani a. Bioorg Med Chem Lett. 2016 Nov 1;26(21):5160-5163. doi: 10.1016/j.bmcl.2016.10.001. Epub 2016 Oct 4. Bioorg Med Chem Lett. 2016. PMID: 27746002 Free article.
Synthesis and biological evaluation of a new class of benzothiazines as neuroprotective agents.
Mancini A, Chelini A, Di Capua A, Castelli L, Brogi S, Paolino M, Giuliani G, Cappelli A, Frosini M, Ricci L, Leonelli E, Giorgi G, Giordani A, Magistretti J, Anzini M. Mancini A, et al. Among authors: giordani a. Eur J Med Chem. 2017 Jan 27;126:614-630. doi: 10.1016/j.ejmech.2016.11.053. Epub 2016 Nov 27. Eur J Med Chem. 2017. PMID: 27923201
122 results