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Gamma-glutamyltransferase, redox regulation and cancer drug resistance.
Curr Opin Pharmacol. 2007 Aug;7(4):360-6. doi: 10.1016/j.coph.2007.04.004. Epub 2007 Jul 5.
Curr Opin Pharmacol. 2007.
PMID: 17613273
Review.
Membrane gamma-glutamyl transferase activity promotes iron-dependent oxidative DNA damage in melanoma cells.
Corti A, Duarte TL, Giommarelli C, De Tata V, Paolicchi A, Jones GD, Pompella A.
Corti A, et al. Among authors: giommarelli c.
Mutat Res. 2009 Oct 2;669(1-2):112-21. doi: 10.1016/j.mrfmmm.2009.05.010. Epub 2009 Jun 6.
Mutat Res. 2009.
PMID: 19505483
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Cellular response to oxidative stress and ascorbic acid in melanoma cells overexpressing gamma-glutamyltransferase.
Giommarelli C, Corti A, Supino R, Favini E, Paolicchi A, Pompella A, Zunino F.
Giommarelli C, et al.
Eur J Cancer. 2008 Mar;44(5):750-9. doi: 10.1016/j.ejca.2008.02.010. Epub 2008 Mar 7.
Eur J Cancer. 2008.
PMID: 18314325
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Gamma-glutamyltransferase-dependent resistance to arsenic trioxide in melanoma cells and cellular sensitization by ascorbic acid.
Giommarelli C, Corti A, Supino R, Favini E, Paolicchi A, Pompella A, Zunino F.
Giommarelli C, et al.
Free Radic Biol Med. 2009 Jun 1;46(11):1516-26. doi: 10.1016/j.freeradbiomed.2009.03.006. Epub 2009 Mar 17.
Free Radic Biol Med. 2009.
PMID: 19298852
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Design, synthesis and anticancer activities of stilbene-coumarin hybrid compounds: Identification of novel proapoptotic agents.
Belluti F, Fontana G, Dal Bo L, Carenini N, Giommarelli C, Zunino F.
Belluti F, et al. Among authors: giommarelli c.
Bioorg Med Chem. 2010 May 15;18(10):3543-50. doi: 10.1016/j.bmc.2010.03.069. Epub 2010 Mar 29.
Bioorg Med Chem. 2010.
PMID: 20409723
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Natural and semisynthetic azaphilones as a new scaffold for Hsp90 inhibitors.
Musso L, Dallavalle S, Merlini L, Bava A, Nasini G, Penco S, Giannini G, Giommarelli C, De Cesare A, Zuco V, Vesci L, Pisano C, Castorina M, Milazzo F, Cervoni ML, Dal Piaz F, De Tommasi N, Zunino F.
Musso L, et al. Among authors: giommarelli c.
Bioorg Med Chem. 2010 Aug 15;18(16):6031-43. doi: 10.1016/j.bmc.2010.06.068. Epub 2010 Jul 1.
Bioorg Med Chem. 2010.
PMID: 20655237
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Isoxazolo(aza)naphthoquinones: a new class of cytotoxic Hsp90 inhibitors.
Bargiotti A, Musso L, Dallavalle S, Merlini L, Gallo G, Ciacci A, Giannini G, Cabri W, Penco S, Vesci L, Castorina M, Milazzo FM, Cervoni ML, Barbarino M, Pisano C, Giommarelli C, Zuco V, De Cesare M, Zunino F.
Bargiotti A, et al. Among authors: giommarelli c.
Eur J Med Chem. 2012 Jul;53:64-75. doi: 10.1016/j.ejmech.2012.03.036. Epub 2012 Mar 28.
Eur J Med Chem. 2012.
PMID: 22538015
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The enhancement of antiproliferative and proapoptotic activity of HDAC inhibitors by curcumin is mediated by Hsp90 inhibition.
Giommarelli C, Zuco V, Favini E, Pisano C, Dal Piaz F, De Tommasi N, Zunino F.
Giommarelli C, et al.
Cell Mol Life Sci. 2010 Mar;67(6):995-1004. doi: 10.1007/s00018-009-0233-x. Epub 2009 Dec 29.
Cell Mol Life Sci. 2010.
PMID: 20039095
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