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KV1.2 channel-specific blocker from Mesobuthus eupeus scorpion venom: Structural basis of selectivity.
Neuropharmacology. 2018 Dec;143:228-238. doi: 10.1016/j.neuropharm.2018.09.030. Epub 2018 Sep 22.
Neuropharmacology. 2018.
PMID: 30248306
Tuning Scorpion Toxin Selectivity: Switching From KV1.1 to KV1.3.
Gigolaev AM, Kuzmenkov AI, Peigneur S, Tabakmakher VM, Pinheiro-Junior EL, Chugunov AO, Efremov RG, Tytgat J, Vassilevski AA.
Gigolaev AM, et al.
Front Pharmacol. 2020 Jul 7;11:1010. doi: 10.3389/fphar.2020.01010. eCollection 2020.
Front Pharmacol. 2020.
PMID: 32733247
Free PMC article.
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Potassium channel blocker crafted by α-hairpinin scaffold engineering.
Tabakmakher VM, Gigolaev AM, Peigneur S, Krylov NA, Tytgat J, Chugunov AO, Vassilevski AA, Efremov RG.
Tabakmakher VM, et al. Among authors: gigolaev am.
Biophys J. 2021 Jun 15;120(12):2471-2481. doi: 10.1016/j.bpj.2021.04.020. Epub 2021 Apr 29.
Biophys J. 2021.
PMID: 33932436
Free PMC article.
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Artificial pore blocker acts specifically on voltage-gated potassium channel isoform KV1.6.
Gigolaev AM, Lushpa VA, Pinheiro-Junior EL, Tabakmakher VM, Peigneur S, Ignatova AA, Feofanov AV, Efremov RG, Mineev KS, Tytgat J, Vassilevski AA.
Gigolaev AM, et al.
J Biol Chem. 2022 Nov;298(11):102467. doi: 10.1016/j.jbc.2022.102467. Epub 2022 Sep 8.
J Biol Chem. 2022.
PMID: 36087839
Free PMC article.
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Scorpion toxins interact with nicotinic acetylcholine receptors.
Kasheverov IE, Oparin PB, Zhmak MN, Egorova NS, Ivanov IA, Gigolaev AM, Nekrasova OV, Serebryakova MV, Kudryavtsev DS, Prokopev NA, Hoang AN, Tsetlin VI, Vassilevski AA, Utkin YN.
Kasheverov IE, et al. Among authors: gigolaev am.
FEBS Lett. 2019 Oct;593(19):2779-2789. doi: 10.1002/1873-3468.13530. Epub 2019 Jul 18.
FEBS Lett. 2019.
PMID: 31276191
Free article.
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Methionine-isoleucine dichotomy at a key position in scorpion toxins inhibiting voltage-gated potassium channels.
Kuzmenkov AI, Gigolaev AM, Pinheiro-Junior EL, Peigneur S, Tytgat J, Vassilevski AA.
Kuzmenkov AI, et al. Among authors: gigolaev am.
Toxicon. 2023 Aug 1;231:107181. doi: 10.1016/j.toxicon.2023.107181. Epub 2023 Jun 8.
Toxicon. 2023.
PMID: 37301298
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