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Structure-Activity Relationships of Cbx7 Inhibitors, Including Selectivity Studies against Other Cbx Proteins.
ACS Omega. 2016 Oct 31;1(4):541-551. doi: 10.1021/acsomega.6b00120. Epub 2016 Oct 12.
ACS Omega. 2016.
PMID: 30023485
Free PMC article.
In Vitro Assessment of Putative PD-1/PD-L1 Inhibitors: Suggestions of an Alternative Mode of Action.
Blevins DJ, Hanley R, Bolduc T, Powell DA, Gignac M, Walker K, Carr MD, Hof F, Wulff JE.
Blevins DJ, et al.
ACS Med Chem Lett. 2019 Jul 2;10(8):1187-1192. doi: 10.1021/acsmedchemlett.9b00221. eCollection 2019 Aug 8.
ACS Med Chem Lett. 2019.
PMID: 31413804
Free PMC article.
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Chromodomain antagonists that target the polycomb-group methyllysine reader protein chromobox homolog 7 (CBX7).
Simhadri C, Daze KD, Douglas SF, Quon TT, Dev A, Gignac MC, Peng F, Heller M, Boulanger MJ, Wulff JE, Hof F.
Simhadri C, et al. Among authors: gignac mc.
J Med Chem. 2014 Apr 10;57(7):2874-83. doi: 10.1021/jm401487x. Epub 2014 Mar 26.
J Med Chem. 2014.
PMID: 24625057
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Selective Inhibition of CBX6: A Methyllysine Reader Protein in the Polycomb Family.
Milosevich N, Gignac MC, McFarlane J, Simhadri C, Horvath S, Daze KD, Croft CS, Dheri A, Quon TT, Douglas SF, Wulff JE, Paci I, Hof F.
Milosevich N, et al. Among authors: gignac mc.
ACS Med Chem Lett. 2015 Dec 7;7(2):139-44. doi: 10.1021/acsmedchemlett.5b00378. eCollection 2016 Feb 11.
ACS Med Chem Lett. 2015.
PMID: 26985288
Free PMC article.
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Robustness of In Vitro Selection Assays of DNA-Encoded Peptidomimetic Ligands to CBX7 and CBX8.
Denton KE, Wang S, Gignac MC, Milosevich N, Hof F, Dykhuizen EC, Krusemark CJ.
Denton KE, et al. Among authors: gignac mc.
SLAS Discov. 2018 Jun;23(5):417-428. doi: 10.1177/2472555217750871. Epub 2018 Jan 8.
SLAS Discov. 2018.
PMID: 29309209
Free PMC article.
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Optimization of Ligands Using Focused DNA-Encoded Libraries To Develop a Selective, Cell-Permeable CBX8 Chromodomain Inhibitor.
Wang S, Denton KE, Hobbs KF, Weaver T, McFarlane JMB, Connelly KE, Gignac MC, Milosevich N, Hof F, Paci I, Musselman CA, Dykhuizen EC, Krusemark CJ.
Wang S, et al. Among authors: gignac mc.
ACS Chem Biol. 2020 Jan 17;15(1):112-131. doi: 10.1021/acschembio.9b00654. Epub 2019 Dec 12.
ACS Chem Biol. 2020.
PMID: 31755685
Free PMC article.
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Aza-amino acid scanning of chromobox homolog 7 (CBX7) ligands.
Traoré M, Gignac M, Doan ND, Hof F, Lubell WD.
Traoré M, et al.
J Pept Sci. 2017 Apr;23(4):266-271. doi: 10.1002/psc.2982. Epub 2017 Feb 21.
J Pept Sci. 2017.
PMID: 28220557
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Pan-specific and partially selective dye-labeled peptidic inhibitors of the polycomb paralog proteins.
Milosevich N, McFarlane J, Gignac MC, Li J, Brown TM, Wilson CR, Devorkin L, Croft CS, Hof R, Paci I, Lum JJ, Hof F.
Milosevich N, et al. Among authors: gignac mc.
Bioorg Med Chem. 2020 Jan 1;28(1):115176. doi: 10.1016/j.bmc.2019.115176. Epub 2019 Nov 9.
Bioorg Med Chem. 2020.
PMID: 31753799
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