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433 results

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Page 1
A novel atypical retinoid endowed with proapoptotic and antitumor activity.
Cincinelli R, Dallavalle S, Merlini L, Penco S, Pisano C, Carminati P, Giannini G, Vesci L, Gaetano C, Illy B, Zuco V, Supino R, Zunino F. Cincinelli R, et al. Among authors: giannini g. J Med Chem. 2003 Mar 13;46(6):909-12. doi: 10.1021/jm025593y. J Med Chem. 2003. PMID: 12620066
Heterocyclic and phenyl double-bond-locked combretastatin analogues possessing potent apoptosis-inducing activity in HL60 and in MDR cell lines.
Simoni D, Grisolia G, Giannini G, Roberti M, Rondanin R, Piccagli L, Baruchello R, Rossi M, Romagnoli R, Invidiata FP, Grimaudo S, Jung MK, Hamel E, Gebbia N, Crosta L, Abbadessa V, Di Cristina A, Dusonchet L, Meli M, Tolomeo M. Simoni D, et al. Among authors: giannini g. J Med Chem. 2005 Feb 10;48(3):723-36. doi: 10.1021/jm049622b. J Med Chem. 2005. PMID: 15689156
Synthesis and structure-activity relationships of a new series of retinoid-related biphenyl-4-ylacrylic acids endowed with antiproliferative and proapoptotic activity.
Cincinelli R, Dallavalle S, Nannei R, Carella S, De Zani D, Merlini L, Penco S, Garattini E, Giannini G, Pisano C, Vesci L, Carminati P, Zuco V, Zanchi C, Zunino F. Cincinelli R, et al. Among authors: giannini g. J Med Chem. 2005 Jul 28;48(15):4931-46. doi: 10.1021/jm049440h. J Med Chem. 2005. PMID: 16033272
Biological and molecular properties of a new alpha(v)beta3/alpha(v)beta5 integrin antagonist.
Belvisi L, Riccioni T, Marcellini M, Vesci L, Chiarucci I, Efrati D, Potenza D, Scolastico C, Manzoni L, Lombardo K, Stasi MA, Orlandi A, Ciucci A, Nico B, Ribatti D, Giannini G, Presta M, Carminati P, Pisano C. Belvisi L, et al. Among authors: giannini g. Mol Cancer Ther. 2005 Nov;4(11):1670-80. doi: 10.1158/1535-7163.MCT-05-0120. Mol Cancer Ther. 2005. PMID: 16275988
Novel combretastatin analogues endowed with antitumor activity.
Simoni D, Romagnoli R, Baruchello R, Rondanin R, Rizzi M, Pavani MG, Alloatti D, Giannini G, Marcellini M, Riccioni T, Castorina M, Guglielmi MB, Bucci F, Carminati P, Pisano C. Simoni D, et al. Among authors: giannini g. J Med Chem. 2006 Jun 1;49(11):3143-52. doi: 10.1021/jm0510732. J Med Chem. 2006. PMID: 16722633
Synthesis and cytotoxic activity of polyamine analogues of camptothecin.
Dallavalle S, Giannini G, Alloatti D, Casati A, Marastoni E, Musso L, Merlini L, Morini G, Penco S, Pisano C, Tinelli S, De Cesare M, Beretta GL, Zunino F. Dallavalle S, et al. Among authors: giannini g. J Med Chem. 2006 Aug 24;49(17):5177-86. doi: 10.1021/jm060285b. J Med Chem. 2006. PMID: 16913706
Synthesis and biological activity of fluorinated combretastatin analogues.
Alloatti D, Giannini G, Cabri W, Lustrati I, Marzi M, Ciacci A, Gallo G, Tinti MO, Marcellini M, Riccioni T, Guglielmi MB, Carminati P, Pisano C. Alloatti D, et al. Among authors: giannini g. J Med Chem. 2008 May 8;51(9):2708-21. doi: 10.1021/jm701362m. Epub 2008 Apr 9. J Med Chem. 2008. PMID: 18396857
433 results