Giacomini E - Search Results

1

The Use of Stilbene Scaffold in Medicinal Chemistry and Multi- Target Drug Design.

Giacomini E, Rupiani S, Guidotti L, Recanatini M, Roberti M. Giacomini E, et al. Curr Med Chem. 2016;23(23):2439-89. doi: 10.2174/0929867323666160517121629. Curr Med Chem. 2016. PMID: 27183980 Review.

2

Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitors.

Rupiani S, Buonfiglio R, Manerba M, Di Ianni L, Vettraino M, Giacomini E, Masetti M, Falchi F, Di Stefano G, Roberti M, Recanatini M. Rupiani S, et al. Among authors: giacomini e. Eur J Med Chem. 2015 Aug 28;101:63-70. doi: 10.1016/j.ejmech.2015.06.028. Epub 2015 Jun 18. Eur J Med Chem. 2015. PMID: 26114812

3

Novel antiproliferative chimeric compounds with marked histone deacetylase inhibitory activity.

Giacomini E, Nebbioso A, Ciotta A, Ianni C, Falchi F, Roberti M, Tolomeo M, Grimaudo S, Cristina AD, Pipitone RM, Altucci L, Recanatini M. Giacomini E, et al. ACS Med Chem Lett. 2014 Jul 8;5(9):973-8. doi: 10.1021/ml5000959. eCollection 2014 Sep 11. ACS Med Chem Lett. 2014. PMID: 25221651 Free PMC article.

4

A ligand-based virtual screening approach to identify small molecules as HERG channel activators.

Giacomini E, Buonfiglio R, Masetti M, Wang Y, Tseng GN, Roberti M, Recanatini M. Giacomini E, et al. Comb Chem High Throughput Screen. 2015;18(3):269-80. doi: 10.2174/1386207318666150305121841. Comb Chem High Throughput Screen. 2015. PMID: 25747449

5

In vitro antileishmanial activity of trans-stilbene and terphenyl compounds.

Castelli G, Bruno F, Vitale F, Roberti M, Colomba C, Giacomini E, Guidotti L, Cascio A, Tolomeo M. Castelli G, et al. Among authors: giacomini e. Exp Parasitol. 2016 Jul;166:1-9. doi: 10.1016/j.exppara.2016.03.007. Epub 2016 Mar 4. Exp Parasitol. 2016. PMID: 26953250

6

Synthesis of natural urolithin M6, a galloflavin mimetic, as a potential inhibitor of lactate dehydrogenase A.

Rupiani S, Guidotti L, Manerba M, Di Ianni L, Giacomini E, Falchi F, Di Stefano G, Roberti M, Recanatini M. Rupiani S, et al. Among authors: giacomini e. Org Biomol Chem. 2016 Nov 22;14(46):10981-10987. doi: 10.1039/c6ob01977c. Org Biomol Chem. 2016. PMID: 27827510

7

Rad51/BRCA2 disruptors inhibit homologous recombination and synergize with olaparib in pancreatic cancer cells.

Roberti M, Schipani F, Bagnolini G, Milano D, Giacomini E, Falchi F, Balboni A, Manerba M, Farabegoli F, De Franco F, Robertson J, Minucci S, Pallavicini I, Di Stefano G, Girotto S, Pellicciari R, Cavalli A. Roberti M, et al. Among authors: giacomini e. Eur J Med Chem. 2019 Mar 1;165:80-92. doi: 10.1016/j.ejmech.2019.01.008. Epub 2019 Jan 10. Eur J Med Chem. 2019. PMID: 30660828

8

Galloflavin (CAS 568-80-9): a novel inhibitor of lactate dehydrogenase.

Manerba M, Vettraino M, Fiume L, Di Stefano G, Sartini A, Giacomini E, Buonfiglio R, Roberti M, Recanatini M. Manerba M, et al. Among authors: giacomini e. ChemMedChem. 2012 Feb 6;7(2):311-7. doi: 10.1002/cmdc.201100471. Epub 2011 Nov 4. ChemMedChem. 2012. PMID: 22052811

9

A natural-like synthetic small molecule impairs bcr-abl signaling cascades and induces megakaryocyte differentiation in erythroleukemia cells.

Turroni S, Tolomeo M, Mamone G, Picariello G, Giacomini E, Brigidi P, Roberti M, Grimaudo S, Pipitone RM, Di Cristina A, Recanatini M. Turroni S, et al. Among authors: giacomini e. PLoS One. 2013;8(2):e57650. doi: 10.1371/journal.pone.0057650. Epub 2013 Feb 27. PLoS One. 2013. PMID: 23460890 Free PMC article.

10

Effects of trans-stilbene and terphenyl compounds on different strains of Leishmania and on cytokines production from infected macrophages.

Bruno F, Castelli G, Vitale F, Giacomini E, Roberti M, Colomba C, Cascio A, Tolomeo M. Bruno F, et al. Among authors: giacomini e. Exp Parasitol. 2018 Jan;184:31-38. doi: 10.1016/j.exppara.2017.11.004. Epub 2017 Nov 14. Exp Parasitol. 2018. PMID: 29154845

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

178 results

Search Page