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Discovery of a Novel Class of Covalent Dual Inhibitors Targeting the Protein Kinases BMX and BTK.
Int J Mol Sci. 2020 Dec 4;21(23):9269. doi: 10.3390/ijms21239269.
Int J Mol Sci. 2020.
PMID: 33291717
Free PMC article.
Development of the First Covalent Monopolar Spindle Kinase 1 (MPS1/TTK) Inhibitor.
M Serafim RA, da Silva Santiago A, Schwalm MP, Hu Z, Dos Reis CV, Takarada JE, Mezzomo P, Massirer KB, Kudolo M, Gerstenecker S, Chaikuad A, Zender L, Knapp S, Laufer S, Couñago RM, Gehringer M.
M Serafim RA, et al. Among authors: gerstenecker s.
J Med Chem. 2022 Feb 24;65(4):3173-3192. doi: 10.1021/acs.jmedchem.1c01165. Epub 2022 Feb 15.
J Med Chem. 2022.
PMID: 35167750
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Discovery of a Potent and Highly Isoform-Selective Inhibitor of the Neglected Ribosomal Protein S6 Kinase Beta 2 (S6K2).
Gerstenecker S, Haarer L, Schröder M, Kudolo M, Schwalm MP, Wydra V, Serafim RAM, Chaikuad A, Knapp S, Laufer S, Gehringer M.
Gerstenecker S, et al.
Cancers (Basel). 2021 Oct 13;13(20):5133. doi: 10.3390/cancers13205133.
Cancers (Basel). 2021.
PMID: 34680283
Free PMC article.
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Protein-Induced Change in Ligand Protonation during Trypsin and Thrombin Binding: Hint on Differences in Selectivity Determinants of Both Proteins?
Ngo K, Collins-Kautz C, Gerstenecker S, Wagner B, Heine A, Klebe G.
Ngo K, et al. Among authors: gerstenecker s.
J Med Chem. 2020 Mar 26;63(6):3274-3289. doi: 10.1021/acs.jmedchem.9b02061. Epub 2020 Feb 24.
J Med Chem. 2020.
PMID: 32011145
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