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A CD3-bispecific molecule targeting P-cadherin demonstrates T cell-mediated regression of established solid tumors in mice.
Cancer Immunol Immunother. 2018 Feb;67(2):247-259. doi: 10.1007/s00262-017-2081-0. Epub 2017 Oct 24.
Cancer Immunol Immunother. 2018.
PMID: 29067496
Free PMC article.
IkappaBalpha kinase inhibitor IKI-1 conferred tumor necrosis factor alpha sensitivity to pancreatic cancer cells and a xenograft tumor model.
Zhang Y, Gavriil M, Lucas J, Mandiyan S, Follettie M, Diesl V, Sum FW, Powell D, Haney S, Abraham R, Arndt K.
Zhang Y, et al. Among authors: gavriil m.
Cancer Res. 2008 Nov 15;68(22):9519-24. doi: 10.1158/0008-5472.CAN-08-1549.
Cancer Res. 2008.
PMID: 19010928
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Specific IKKbeta inhibitor IV blocks Streptonigrin-induced NF-kappaB activity and potentiates its cytotoxic effect on cancer cells.
Gavriil M, Tsao CC, Mandiyan S, Arndt K, Abraham R, Zhang Y.
Gavriil M, et al.
Mol Carcinog. 2009 Aug;48(8):678-84. doi: 10.1002/mc.20550.
Mol Carcinog. 2009.
PMID: 19444813
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Combination therapy for treating breast cancer using antiestrogen, ERA-923, and the mammalian target of rapamycin inhibitor, temsirolimus.
Sadler TM, Gavriil M, Annable T, Frost P, Greenberger LM, Zhang Y.
Sadler TM, et al. Among authors: gavriil m.
Endocr Relat Cancer. 2006 Sep;13(3):863-73. doi: 10.1677/erc.1.01170.
Endocr Relat Cancer. 2006.
PMID: 16954435
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Synthesis and biological evaluation of tricyclic anilinopyrimidines as IKKbeta inhibitors.
Crombie AL, Sum FW, Powell DW, Hopper DW, Torres N, Berger DM, Zhang Y, Gavriil M, Sadler TM, Arndt K.
Crombie AL, et al. Among authors: gavriil m.
Bioorg Med Chem Lett. 2010 Jun 15;20(12):3821-5. doi: 10.1016/j.bmcl.2010.04.022. Epub 2010 Apr 18.
Bioorg Med Chem Lett. 2010.
PMID: 20471256
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2-Hydroxyglutarate modulates histone methylation at specific loci and alters gene expression via Rph1 inhibition.
Gavriil M, Proietto M, Paczia N, Ginolhac A, Halder R, Valceschini E, Sauter T, Linster CL, Sinkkonen L.
Gavriil M, et al.
Life Sci Alliance. 2023 Nov 27;7(2):e202302333. doi: 10.26508/lsa.202302333. Print 2024 Feb.
Life Sci Alliance. 2023.
PMID: 38011998
Free PMC article.
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ATG5 and ATG7 Expression Levels Are Reduced in Cutaneous Melanoma and Regulated by NRF1.
Frangež Ž, Gérard D, He Z, Gavriil M, Fernández-Marrero Y, Seyed Jafari SM, Hunger RE, Lucarelli P, Yousefi S, Sauter T, Sinkkonen L, Simon HU.
Frangež Ž, et al. Among authors: gavriil m.
Front Oncol. 2021 Aug 12;11:721624. doi: 10.3389/fonc.2021.721624. eCollection 2021.
Front Oncol. 2021.
PMID: 34458153
Free PMC article.
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DNA methylation profiling implicates exposure to PCBs in the pathogenesis of B-cell chronic lymphocytic leukemia.
Georgiadis P, Gavriil M, Rantakokko P, Ladoukakis E, Botsivali M, Kelly RS, Bergdahl IA, Kiviranta H, Vermeulen RCH, Spaeth F, Hebbels DGAJ, Kleinjans JCS, de Kok TMCM, Palli D, Vineis P, Kyrtopoulos SA; EnviroGenomarkers consortium.
Georgiadis P, et al. Among authors: gavriil m.
Environ Int. 2019 May;126:24-36. doi: 10.1016/j.envint.2019.01.068. Epub 2019 Feb 15.
Environ Int. 2019.
PMID: 30776747
Free PMC article.
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