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New Phosphoramidates Containing Selenium as Leishmanicidal Agents.
Antimicrob Agents Chemother. 2021 Sep 17;65(10):e0059021. doi: 10.1128/AAC.00590-21. Epub 2021 Aug 2.
Antimicrob Agents Chemother. 2021.
PMID: 34339279
Free PMC article.
Pyridazino-pyrrolo-quinoxalinium salts as highly potent and selective leishmanicidal agents targeting trypanothione reductase.
de Lucio H, García-Marín J, Sánchez-Alonso P, García-Soriano JC, Toro MÁ, Vaquero JJ, Gago F, Alajarín R, Jiménez-Ruiz A.
de Lucio H, et al. Among authors: garcia soriano jc.
Eur J Med Chem. 2022 Jan 5;227:113915. doi: 10.1016/j.ejmech.2021.113915. Epub 2021 Oct 15.
Eur J Med Chem. 2022.
PMID: 34695777
Free article.
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Efficient Dimerization Disruption of Leishmania infantum Trypanothione Reductase by Triazole-phenyl-thiazoles.
Revuelto A, de Lucio H, García-Soriano JC, Sánchez-Murcia PA, Gago F, Jiménez-Ruiz A, Camarasa MJ, Velázquez S.
Revuelto A, et al. Among authors: garcia soriano jc.
J Med Chem. 2021 May 13;64(9):6137-6160. doi: 10.1021/acs.jmedchem.1c00206. Epub 2021 May 4.
J Med Chem. 2021.
PMID: 33945281
Free PMC article.
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Identification of L. infantum trypanothione synthetase inhibitors with leishmanicidal activity from a (non-biased) in-house chemical library.
Alcón-Calderón M, de Lucio H, García-Soriano JC, Revuelto A, de Castro S, López-Gutiérrez C, San-Félix A, Quesada E, Gago F, Camarasa MJ, Jiménez-Ruiz A, Velázquez S.
Alcón-Calderón M, et al. Among authors: garcia soriano jc.
Eur J Med Chem. 2022 Dec 5;243:114675. doi: 10.1016/j.ejmech.2022.114675. Epub 2022 Aug 18.
Eur J Med Chem. 2022.
PMID: 36075146
Free article.
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Small Molecule-Peptide Conjugates as Dimerization Inhibitors of Leishmania infantum Trypanothione Disulfide Reductase.
Revuelto A, López-Martín I, de Lucio H, García-Soriano JC, Zanda N, de Castro S, Gago F, Jiménez-Ruiz A, Velázquez S, Camarasa MJ.
Revuelto A, et al. Among authors: garcia soriano jc.
Pharmaceuticals (Basel). 2021 Jul 17;14(7):689. doi: 10.3390/ph14070689.
Pharmaceuticals (Basel). 2021.
PMID: 34358115
Free PMC article.
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Identification of 1,2,3-triazolium salt-based inhibitors of Leishmania infantum trypanothione disulfide reductase with enhanced antileishmanial potency in cellulo and increased selectivity.
de Lucio H, Revuelto A, Carriles AA, de Castro S, García-González S, García-Soriano JC, Alcón-Calderón M, Sánchez-Murcia PA, Hermoso JA, Gago F, Camarasa MJ, Jiménez-Ruiz A, Velázquez S.
de Lucio H, et al. Among authors: garcia soriano jc.
Eur J Med Chem. 2022 Dec 15;244:114878. doi: 10.1016/j.ejmech.2022.114878. Epub 2022 Oct 29.
Eur J Med Chem. 2022.
PMID: 36332553
Free article.
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