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Histone acetyltransferase inhibitor CPTH6 preferentially targets lung cancer stem-like cells.
Di Martile M, Desideri M, De Luca T, Gabellini C, Buglioni S, Eramo A, Sette G, Milella M, Rotili D, Mai A, Carradori S, Secci D, De Maria R, Del Bufalo D, Trisciuoglio D. Di Martile M, et al. Among authors: gabellini c. Oncotarget. 2016 Mar 8;7(10):11332-48. doi: 10.18632/oncotarget.7238. Oncotarget. 2016. PMID: 26870991 Free PMC article.
CPTH6, a thiazole derivative, induces histone hypoacetylation and apoptosis in human leukemia cells.
Trisciuoglio D, Ragazzoni Y, Pelosi A, Desideri M, Carradori S, Gabellini C, Maresca G, Nescatelli R, Secci D, Bolasco A, Bizzarri B, Cavaliere C, D'Agnano I, Filetici P, Ricci-Vitiani L, Rizzo MG, Del Bufalo D. Trisciuoglio D, et al. Among authors: gabellini c. Clin Cancer Res. 2012 Jan 15;18(2):475-86. doi: 10.1158/1078-0432.CCR-11-0579. Epub 2011 Nov 8. Clin Cancer Res. 2012. PMID: 22068659
Inhibition of lysine acetyltransferases impairs tumor angiogenesis acting on both endothelial and tumor cells.
Di Martile M, Gabellini C, Desideri M, Matraxia M, Farini V, Valentini E, Carradori S, Ercolani C, Buglioni S, Secci D, Andreazzoli M, Del Bufalo D, Trisciuoglio D. Di Martile M, et al. Among authors: gabellini c. J Exp Clin Cancer Res. 2020 Jun 5;39(1):103. doi: 10.1186/s13046-020-01604-z. J Exp Clin Cancer Res. 2020. PMID: 32498717 Free PMC article.
The thiazole derivative CPTH6 impairs autophagy.
Ragazzoni Y, Desideri M, Gabellini C, De Luca T, Carradori S, Secci D, Nescatelli R, Candiloro A, Condello M, Meschini S, Del Bufalo D, Trisciuoglio D. Ragazzoni Y, et al. Among authors: gabellini c. Cell Death Dis. 2013 Mar 7;4(3):e524. doi: 10.1038/cddis.2013.53. Cell Death Dis. 2013. PMID: 23470531 Free PMC article.
BCL-XL overexpression promotes tumor progression-associated properties.
Trisciuoglio D, Tupone MG, Desideri M, Di Martile M, Gabellini C, Buglioni S, Pallocca M, Alessandrini G, D'Aguanno S, Del Bufalo D. Trisciuoglio D, et al. Among authors: gabellini c. Cell Death Dis. 2017 Dec 13;8(12):3216. doi: 10.1038/s41419-017-0055-y. Cell Death Dis. 2017. PMID: 29238043 Free PMC article.
41 results