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Development of Small-Molecule Anti-HIV-1 Agents Targeting HIV-1 Capsid Proteins.
Kobayakawa T, Yokoyama M, Tsuji K, Boku S, Kurakami M, Fujino M, Ishii T, Miura Y, Nishimura S, Shinohara K, Yamamoto K, Bolah P, Kotani O, Murakami T, Sato H, Tamamura H. Kobayakawa T, et al. Among authors: fujino m. Chem Pharm Bull (Tokyo). 2024;72(1):41-47. doi: 10.1248/cpb.c23-00618. Chem Pharm Bull (Tokyo). 2024. PMID: 38171903 Free article.
Exploratory studies on CA-15L, an anti-HIV active HIV-1 capsid fragment.
Tsuji K, Owusu KB, Kobayakawa T, Wang R, Fujino M, Kaneko M, Yamamoto N, Murakami T, Tamamura H. Tsuji K, et al. Among authors: fujino m. Bioorg Med Chem. 2020 Jun 1;28(11):115488. doi: 10.1016/j.bmc.2020.115488. Epub 2020 Apr 8. Bioorg Med Chem. 2020. PMID: 32305183
Potent leads based on CA-19L, an anti-HIV active HIV-1 capsid fragment.
Tsuji K, Wang R, Kobayakawa T, Owusu KB, Fujino M, Kaneko M, Yamamoto N, Murakami T, Tamamura H. Tsuji K, et al. Among authors: fujino m. Bioorg Med Chem. 2021 Jan 15;30:115923. doi: 10.1016/j.bmc.2020.115923. Epub 2020 Dec 7. Bioorg Med Chem. 2021. PMID: 33316719
Small-Molecule Anti-HIV-1 Agents Based on HIV-1 Capsid Proteins.
Kobayakawa T, Yokoyama M, Tsuji K, Fujino M, Kurakami M, Boku S, Nakayama M, Kaneko M, Ohashi N, Kotani O, Murakami T, Sato H, Tamamura H. Kobayakawa T, et al. Among authors: fujino m. Biomolecules. 2021 Feb 3;11(2):208. doi: 10.3390/biom11020208. Biomolecules. 2021. PMID: 33546092 Free PMC article.
Low-molecular-weight anti-HIV-1 agents targeting HIV-1 capsid proteins.
Kobayakawa T, Yokoyama M, Tsuji K, Fujino M, Kurakami M, Onishi T, Boku S, Ishii T, Miura Y, Shinohara K, Kishihara Y, Ohashi N, Kotani O, Murakami T, Sato H, Tamamura H. Kobayakawa T, et al. Among authors: fujino m. RSC Adv. 2023 Jan 12;13(3):2156-2167. doi: 10.1039/d2ra06837k. eCollection 2023 Jan 6. RSC Adv. 2023. PMID: 36712613 Free PMC article.
Anti-HIV-1 peptide derivatives based on the HIV-1 Co-receptor CXCR4.
Hashimoto C, Nomura W, Narumi T, Fujino M, Tsutsumi H, Haseyama M, Yamamoto N, Murakami T, Tamamura H. Hashimoto C, et al. Among authors: fujino m. ChemMedChem. 2013 Oct;8(10):1668-72. doi: 10.1002/cmdc.201300289. Epub 2013 Aug 23. ChemMedChem. 2013. PMID: 24039179
CXCR4-derived synthetic peptides inducing anti-HIV-1 antibodies.
Hashimoto C, Nomura W, Narumi T, Fujino M, Nakahara T, Yamamoto N, Murakami T, Tamamura H. Hashimoto C, et al. Among authors: fujino m. Bioorg Med Chem. 2013 Nov 15;21(22):6878-85. doi: 10.1016/j.bmc.2013.09.037. Epub 2013 Sep 21. Bioorg Med Chem. 2013. PMID: 24119449
Bivalent HIV-1 fusion inhibitors based on peptidomimetics.
Kobayakawa T, Ebihara K, Tsuji K, Kawada T, Fujino M, Honda Y, Ohashi N, Murakami T, Tamamura H. Kobayakawa T, et al. Among authors: fujino m. Bioorg Med Chem. 2020 Dec 15;28(24):115812. doi: 10.1016/j.bmc.2020.115812. Epub 2020 Oct 9. Bioorg Med Chem. 2020. PMID: 33157478
951 results