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2016 | 1 |
2018 | 1 |
2019 | 1 |
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Biological Characterization of 8-Cyclopropyl-2-(pyridin-3-yl)thiazolo[5,4-f]quinazolin-9(8H)-one, a Promising Inhibitor of DYRK1A.
Pharmaceuticals (Basel). 2019 Dec 17;12(4):185. doi: 10.3390/ph12040185.
Pharmaceuticals (Basel). 2019.
PMID: 31861110
Free PMC article.
Development of Kinase Inhibitors via Metal-Catalyzed C⁻H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies.
Couly F, Harari M, Dubouilh-Benard C, Bailly L, Petit E, Diharce J, Bonnet P, Meijer L, Fruit C, Besson T.
Couly F, et al.
Molecules. 2018 Aug 29;23(9):2181. doi: 10.3390/molecules23092181.
Molecules. 2018.
PMID: 30158487
Free PMC article.
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Pd-Catalyzed and Copper Assisted Regioselective Sequential C2 and C7 Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one with Aryl Halides.
Harari M, Couly F, Fruit C, Besson T.
Harari M, et al. Among authors: couly f.
Org Lett. 2016 Jul 1;18(13):3282-5. doi: 10.1021/acs.orglett.6b01552. Epub 2016 Jun 17.
Org Lett. 2016.
PMID: 27314437
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