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Combined SRPK and AKT pharmacological inhibition is synergistic in T-cell acute lymphoblastic leukemia cells.
Siqueira RP, Caetano MMM, de Souza LÂ, Dos Passos PMS, Simaroli NB, Barros MVA, de Souza APM, de Oliveira LL, Silva-Júnior A, Fietto JLR, Teixeira RR, Teixeira FR, Bressan GC. Siqueira RP, et al. Among authors: fietto jlr. Toxicol In Vitro. 2020 Jun;65:104777. doi: 10.1016/j.tiv.2020.104777. Epub 2020 Jan 18. Toxicol In Vitro. 2020. PMID: 31962201 Free article.
Trypanosoma cruzi nucleoside triphosphate diphosphohydrolase 1 (TcNTPDase-1) biochemical characterization, immunolocalization and possible role in host cell adhesion.
Mariotini-Moura C, Silva e Bastos M, de Castro FF, Trindade ML, Vasconcellos Rde S, Neves-do-Valle MA, Moreira BP, Santos Rde F, de Oliveira CM, Cunha LC, Souto XM, Bressan GC, Silva-Júnior A, Baqui MM, Bahia MT, de Almeida MR, Meyer-Fernandes JR, Fietto JL. Mariotini-Moura C, et al. Acta Trop. 2014 Feb;130:140-7. doi: 10.1016/j.actatropica.2013.11.008. Epub 2013 Nov 19. Acta Trop. 2014. PMID: 24269744 Free article.
Leishmania infantum ecto-nucleoside triphosphate diphosphohydrolase-2 is an apyrase involved in macrophage infection and expressed in infected dogs.
Vasconcellos Rde S, Mariotini-Moura C, Gomes RS, Serafim TD, Firmino Rde C, Silva E Bastos M, Castro FF, Oliveira CM, Borges-Pereira L, de Souza AC, de Souza RF, Gómez GA, Pinheiro Ada C, Maciel TE, Silva-Júnior A, Bressan GC, Almeida MR, Baqui MM, Afonso LC, Fietto JL. Vasconcellos Rde S, et al. PLoS Negl Trop Dis. 2014 Nov 13;8(11):e3309. doi: 10.1371/journal.pntd.0003309. eCollection 2014 Nov. PLoS Negl Trop Dis. 2014. PMID: 25393008 Free PMC article.
Potential Antileukemia Effect and Structural Analyses of SRPK Inhibition by N-(2-(Piperidin-1-yl)-5-(Trifluoromethyl)Phenyl)Isonicotinamide (SRPIN340).
Siqueira RP, Barbosa Éde A, Polêto MD, Righetto GL, Seraphim TV, Salgado RL, Ferreira JG, Barros MV, de Oliveira LL, Laranjeira AB, Almeida MR, Júnior AS, Fietto JL, Kobarg J, de Oliveira EB, Teixeira RR, Borges JC, Yunes JA, Bressan GC. Siqueira RP, et al. PLoS One. 2015 Aug 5;10(8):e0134882. doi: 10.1371/journal.pone.0134882. eCollection 2015. PLoS One. 2015. PMID: 26244849 Free PMC article.
Splicing Regulators and Their Roles in Cancer Biology and Therapy.
da Silva MR, Moreira GA, Gonçalves da Silva RA, de Almeida Alves Barbosa É, Pais Siqueira R, Teixera RR, Almeida MR, Silva Júnior A, Fietto JL, Bressan GC. da Silva MR, et al. Biomed Res Int. 2015;2015:150514. doi: 10.1155/2015/150514. Epub 2015 Jul 26. Biomed Res Int. 2015. PMID: 26273588 Free PMC article. Review.
Trifluoromethyl arylamides with antileukemia effect and intracellular inhibitory activity over serine/arginine-rich protein kinases (SRPKs).
Siqueira RP, Barros MVA, Barbosa ÉAA, Onofre TS, Gonçalves VHS, Pereira HS, Silva Júnior A, de Oliveira LL, Almeida MR, Fietto JLR, Teixeira RR, Bressan GC. Siqueira RP, et al. Among authors: fietto jlr. Eur J Med Chem. 2017 Jul 7;134:97-109. doi: 10.1016/j.ejmech.2017.03.078. Epub 2017 Mar 31. Eur J Med Chem. 2017. PMID: 28407594
68 results