Ferorelli S - Search Results

1

Translational impact of novel widely pharmacological characterized mofezolac-derived COX-1 inhibitors combined with bortezomib on human multiple myeloma cell lines viability.

Pati ML, Vitale P, Ferorelli S, Iaselli M, Miciaccia M, Boccarelli A, Di Mauro GD, Fortuna CG, Souza Domingos TF, Rodrigues Pereira da Silva LC, de Pádula M, Cabral LM, Sathler PC, Vacca A, Scilimati A, Perrone MG. Pati ML, et al. Among authors: ferorelli s. Eur J Med Chem. 2019 Feb 15;164:59-76. doi: 10.1016/j.ejmech.2018.12.029. Epub 2018 Dec 15. Eur J Med Chem. 2019. PMID: 30590258

2

4-(tetralin-1-yl)- and 4-(naphthalen-1-yl)alkyl derivatives of 1-cyclohexylpiperazine as sigma receptor ligands with agonist sigma2 activity.

Berardi F, Ferorelli S, Abate C, Colabufo NA, Contino M, Perrone R, Tortorella V. Berardi F, et al. Among authors: ferorelli s. J Med Chem. 2004 Apr 22;47(9):2308-17. doi: 10.1021/jm031026e. J Med Chem. 2004. PMID: 15084129

3

Methyl substitution on the piperidine ring of N-[omega-(6-methoxynaphthalen-1-yl)alkyl] derivatives as a probe for selective binding and activity at the sigma(1) receptor.

Berardi F, Ferorelli S, Abate C, Pedone MP, Colabufo NA, Contino M, Perrone R. Berardi F, et al. Among authors: ferorelli s. J Med Chem. 2005 Dec 29;48(26):8237-44. doi: 10.1021/jm050654o. J Med Chem. 2005. PMID: 16366605

4

Novel 4-(4-aryl)cyclohexyl-1-(2-pyridyl)piperazines as Delta(8)-Delta(7) sterol isomerase (emopamil binding protein) selective ligands with antiproliferative activity.

Berardi F, Abate C, Ferorelli S, de Robertis AF, Leopoldo M, Colabufo NA, Niso M, Perrone R. Berardi F, et al. Among authors: ferorelli s. J Med Chem. 2008 Dec 11;51(23):7523-31. doi: 10.1021/jm800965b. J Med Chem. 2008. PMID: 19053780

5

Exploring the importance of piperazine N-atoms for sigma(2) receptor affinity and activity in a series of analogs of 1-cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28).

Berardi F, Abate C, Ferorelli S, Uricchio V, Colabufo NA, Niso M, Perrone R. Berardi F, et al. Among authors: ferorelli s. J Med Chem. 2009 Dec 10;52(23):7817-28. doi: 10.1021/jm9007505. J Med Chem. 2009. PMID: 19842660

6

Arylamides hybrids of two high-affinity σ2 receptor ligands as tools for the development of PET radiotracers.

Abate C, Ferorelli S, Contino M, Marottoli R, Colabufo NA, Perrone R, Berardi F. Abate C, et al. Among authors: ferorelli s. Eur J Med Chem. 2011 Sep;46(9):4733-41. doi: 10.1016/j.ejmech.2011.05.057. Epub 2011 May 30. Eur J Med Chem. 2011. PMID: 21684636

7

Synthesis and binding assays of novel 3,3-dimethylpiperidine derivatives with various lipophilicities as σ₁ receptor ligands.

Ferorelli S, Abate C, Pedone MP, Colabufo NA, Contino M, Perrone R, Berardi F. Ferorelli S, et al. Bioorg Med Chem. 2011 Dec 15;19(24):7612-22. doi: 10.1016/j.bmc.2011.10.023. Epub 2011 Oct 17. Bioorg Med Chem. 2011. PMID: 22075234

8

Deconstruction of 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline moiety to separate P-glycoprotein (P-gp) activity from σ2 receptor affinity in mixed P-gp/σ2 receptor agents.

Pati ML, Abate C, Contino M, Ferorelli S, Luisi R, Carroccia L, Niso M, Berardi F. Pati ML, et al. Among authors: ferorelli s. Eur J Med Chem. 2015 Jan 7;89:691-700. doi: 10.1016/j.ejmech.2014.11.001. Epub 2014 Nov 4. Eur J Med Chem. 2015. PMID: 25462276

9

Isoxazole-Based-Scaffold Inhibitors Targeting Cyclooxygenases (COXs).

Perrone MG, Vitale P, Panella A, Ferorelli S, Contino M, Lavecchia A, Scilimati A. Perrone MG, et al. Among authors: ferorelli s. ChemMedChem. 2016 Jun 6;11(11):1172-87. doi: 10.1002/cmdc.201500439. Epub 2016 May 2. ChemMedChem. 2016. PMID: 27136372

10

Structural basis for selective inhibition of Cyclooxygenase-1 (COX-1) by diarylisoxazoles mofezolac and 3-(5-chlorofuran-2-yl)-5-methyl-4-phenylisoxazole (P6).

Cingolani G, Panella A, Perrone MG, Vitale P, Di Mauro G, Fortuna CG, Armen RS, Ferorelli S, Smith WL, Scilimati A. Cingolani G, et al. Among authors: ferorelli s. Eur J Med Chem. 2017 Sep 29;138:661-668. doi: 10.1016/j.ejmech.2017.06.045. Epub 2017 Jun 24. Eur J Med Chem. 2017. PMID: 28710965 Free PMC article.

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