Fernández-Bachiller MI - Search Results

1

Probing Factor Xa Protein-Ligand Interactions: Accurate Free Energy Calculations and Experimental Validations of Two Series of High-Affinity Ligands.

Fernández-Bachiller MI, Hwang S, Schembri ME, Lindemann P, Guberman M, Herziger S, Specker E, Matter H, Will DW, Czech J, Wagner M, Bauer A, Schreuder H, Ritter K, Urmann M, Wehner V, Sun H, Nazaré M. Fernández-Bachiller MI, et al. J Med Chem. 2022 Oct 13;65(19):13013-13028. doi: 10.1021/acs.jmedchem.2c00865. Epub 2022 Sep 30. J Med Chem. 2022. PMID: 36178213

2

Alzheimer's disease: identification and development of β-secretase (BACE-1) binding fragments and inhibitors by dynamic ligation screening (DLS).

Fernández-Bachiller MI, Horatscheck A, Lisurek M, Rademann J. Fernández-Bachiller MI, et al. ChemMedChem. 2013 Jul;8(7):1041-56. doi: 10.1002/cmdc.201300078. Epub 2013 Jun 11. ChemMedChem. 2013. PMID: 23757181

3

Mapping Protein-Protein Interactions of the Resistance-Related Bacterial Zeta Toxin-Epsilon Antitoxin Complex (ε₂ζ₂) with High Affinity Peptide Ligands Using Fluorescence Polarization.

Fernández-Bachiller MI, Brzozowska I, Odolczyk N, Zielenkiewicz U, Zielenkiewicz P, Rademann J. Fernández-Bachiller MI, et al. Toxins (Basel). 2016 Jul 16;8(7):222. doi: 10.3390/toxins8070222. Toxins (Basel). 2016. PMID: 27438853 Free PMC article.

4

Chemoselective Wittig and Michael ligations of unprotected peptidyl phosphoranes in water furnish potent inhibitors of caspase-3.

Holland-Nell K, Fernández-Bachiller MI, Ahsanullah, Rademann J. Holland-Nell K, et al. Among authors: fernandez bachiller mi. Org Lett. 2014 Sep 5;16(17):4428-31. doi: 10.1021/ol501910x. Epub 2014 Aug 20. Org Lett. 2014. PMID: 25141292

5

New tacrine-4-oxo-4H-chromene hybrids as multifunctional agents for the treatment of Alzheimer's disease, with cholinergic, antioxidant, and β-amyloid-reducing properties.

Fernández-Bachiller MI, Pérez C, Monjas L, Rademann J, Rodríguez-Franco MI. Fernández-Bachiller MI, et al. J Med Chem. 2012 Feb 9;55(3):1303-17. doi: 10.1021/jm201460y. Epub 2012 Jan 27. J Med Chem. 2012. PMID: 22243648

6

Syntheses of defined sulfated oligohyaluronans reveal structural effects, diversity and thermodynamics of GAG-protein binding.

Köhling S, Blaszkiewicz J, Ruiz-Gómez G, Fernández-Bachiller MI, Lemmnitzer K, Panitz N, Beck-Sickinger AG, Schiller J, Pisabarro MT, Rademann J. Köhling S, et al. Among authors: fernandez bachiller mi. Chem Sci. 2018 Nov 1;10(3):866-878. doi: 10.1039/c8sc03649g. eCollection 2019 Jan 21. Chem Sci. 2018. PMID: 30774881 Free PMC article.

7

Tacrine-melatonin hybrids as multifunctional agents for Alzheimer's disease, with cholinergic, antioxidant, and neuroprotective properties.

Fernández-Bachiller MI, Pérez C, Campillo NE, Páez JA, González-Muñoz GC, Usán P, García-Palomero E, López MG, Villarroya M, García AG, Martínez A, Rodríguez-Franco MI. Fernández-Bachiller MI, et al. ChemMedChem. 2009 May;4(5):828-41. doi: 10.1002/cmdc.200800414. ChemMedChem. 2009. PMID: 19308922

8

Novel tacrine-melatonin hybrids as dual-acting drugs for Alzheimer disease, with improved acetylcholinesterase inhibitory and antioxidant properties.

Rodríguez-Franco MI, Fernández-Bachiller MI, Pérez C, Hernández-Ledesma B, Bartolomé B. Rodríguez-Franco MI, et al. J Med Chem. 2006 Jan 26;49(2):459-62. doi: 10.1021/jm050746d. J Med Chem. 2006. PMID: 16420031

9

Novel tacrine-8-hydroxyquinoline hybrids as multifunctional agents for the treatment of Alzheimer's disease, with neuroprotective, cholinergic, antioxidant, and copper-complexing properties.

Fernández-Bachiller MI, Pérez C, González-Muñoz GC, Conde S, López MG, Villarroya M, García AG, Rodríguez-Franco MI. Fernández-Bachiller MI, et al. J Med Chem. 2010 Jul 8;53(13):4927-37. doi: 10.1021/jm100329q. J Med Chem. 2010. PMID: 20545360

10

Design and synthesis of N-benzylpiperidine-purine derivatives as new dual inhibitors of acetyl- and butyrylcholinesterase.

Rodríguez-Franco MI, Fernández-Bachiller MI, Pérez C, Castro A, Martínez A. Rodríguez-Franco MI, et al. Bioorg Med Chem. 2005 Dec 15;13(24):6795-802. doi: 10.1016/j.bmc.2005.07.019. Epub 2005 Sep 23. Bioorg Med Chem. 2005. PMID: 16183292

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