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Structural elucidation of the DFG-Asp in and DFG-Asp out states of TAM kinases and insight into the selectivity of their inhibitors.
Molecules. 2014 Oct 10;19(10):16223-39. doi: 10.3390/molecules191016223.
Molecules. 2014.
PMID: 25310149
Free PMC article.
Recent progress in the design, study, and development of c-Jun N-terminal kinase inhibitors as anticancer agents.
Messoussi A, Feneyrolles C, Bros A, Deroide A, Daydé-Cazals B, Chevé G, Van Hijfte N, Fauvel B, Bougrin K, Yasri A.
Messoussi A, et al. Among authors: feneyrolles c.
Chem Biol. 2014 Nov 20;21(11):1433-43. doi: 10.1016/j.chembiol.2014.09.007. Epub 2014 Oct 16.
Chem Biol. 2014.
PMID: 25442375
Review.
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Axl kinase as a key target for oncology: focus on small molecule inhibitors.
Feneyrolles C, Spenlinhauer A, Guiet L, Fauvel B, Daydé-Cazals B, Warnault P, Chevé G, Yasri A.
Feneyrolles C, et al.
Mol Cancer Ther. 2014 Sep;13(9):2141-8. doi: 10.1158/1535-7163.MCT-13-1083. Epub 2014 Aug 19.
Mol Cancer Ther. 2014.
PMID: 25139999
Review.
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Discovering novel 7-azaindole-based series as potent AXL kinase inhibitors.
Feneyrolles C, Guiet L, Singer M, Van Hijfte N, Daydé-Cazals B, Fauvel B, Chevé G, Yasri A.
Feneyrolles C, et al.
Bioorg Med Chem Lett. 2017 Feb 15;27(4):862-866. doi: 10.1016/j.bmcl.2017.01.015. Epub 2017 Jan 9.
Bioorg Med Chem Lett. 2017.
PMID: 28094183
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Rational Design, Synthesis, and Biological Evaluation of 7-Azaindole Derivatives as Potent Focused Multi-Targeted Kinase Inhibitors.
Daydé-Cazals B, Fauvel B, Singer M, Feneyrolles C, Bestgen B, Gassiot F, Spenlinhauer A, Warnault P, Van Hijfte N, Borjini N, Chevé G, Yasri A.
Daydé-Cazals B, et al. Among authors: feneyrolles c.
J Med Chem. 2016 Apr 28;59(8):3886-905. doi: 10.1021/acs.jmedchem.6b00087. Epub 2016 Apr 15.
J Med Chem. 2016.
PMID: 27010810
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